FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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3 compounds in matrix 5 best compound-target hits listed 4 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T03T11T16T18
ulfkktlib_1655
[H]N(Cc1ccccn1)C(=O)c1cnc(-c2ccccc2)nc1[C@H]1CC(=O)N(c2ccccc2)C1
0.872 0.852 2 0.87 0.83
ulfkktlib_165
[H]N(CCc1cn([H])c2ccccc12)C(=O)[C@H](Cc1cn([H])c2ccccc12)[N+]([H])([H])CCCC
0.850 0.837 2 0.85 0.82
ulfkktlib_1652
[H]N(C(=O)c1cnc(-c2ccccc2)nc1[C@@H]1CC(=O)N(c2ccccc2)C1)C1CCCCC1
0.820 0.820 1 0.82

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
ulfkktlib_1655
[H]N(Cc1ccccn1)C(=O)c1cnc(-c2ccccc2)nc1[C@H]1CC(=O)N(c2ccccc2)C1
T11
native IFP available
T11
dockmulti_91311c650f2e_T11
0.872 1.000 0.636 native_similarity final_rank_score -17.3697 -0.646662 13 4 Pose
ulfkktlib_165
[H]N(CCc1cn([H])c2ccccc12)C(=O)[C@H](Cc1cn([H])c2ccccc12)[N+]([H])([H])CCCC
T11
native IFP available
T11
dockmulti_91311c650f2e_T11
0.850 1.000 0.573 native_similarity final_rank_score -20.3852 -0.809111 18 5 Pose
ulfkktlib_1655
[H]N(Cc1ccccn1)C(=O)c1cnc(-c2ccccc2)nc1[C@H]1CC(=O)N(c2ccccc2)C1
T18
native IFP available
T18
dockmulti_91311c650f2e_T18
0.831 1.000 0.516 native_similarity final_rank_score -18.4771 -0.524252 11 2 Pose
ulfkktlib_165
[H]N(CCc1cn([H])c2ccccc12)C(=O)[C@H](Cc1cn([H])c2ccccc12)[N+]([H])([H])CCCC
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.823 1.000 0.495 native_similarity final_rank_score -14.4088 -0.736052 19 4 Pose
ulfkktlib_1652
[H]N(C(=O)c1cnc(-c2ccccc2)nc1[C@@H]1CC(=O)N(c2ccccc2)C1)C1CCCCC1
T03
native IFP available
T03
dockmulti_91311c650f2e_T03
0.820 1.000 0.486 native_similarity final_rank_score -23.0451 -0.682003 18 1 Pose