FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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3 compounds in matrix 6 best compound-target hits listed 6 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T03T09T16T18T20
Z57985071
[H]N(C(=O)C[C@@H]1S/C(=N\c2ccccc2)N(CCc2cn([H])c3ccccc23)C1=O)c1ccccc1F
0.936 0.936 1 0.94
Z57985071
[H]N(C(=O)C[C@H]1S/C(=N/c2ccccc2)N(CCc2cn([H])c3ccccc23)C1=O)c1ccccc1F
0.854 0.812 3 0.80 0.85 0.78
Z57985071
[H]N(C(=O)C[C@@H]1S/C(=N/c2ccccc2)N(CCc2cn([H])c3ccccc23)C1=O)c1ccccc1F
0.843 0.831 2 0.82 0.84

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z57985071
[H]N(C(=O)C[C@@H]1S/C(=N\c2ccccc2)N(CCc2cn([H])c3ccccc23)C1=O)c1ccccc1F
T20
native IFP available
T20
dockmulti_91311c650f2e_T20
0.936 1.000 0.817 native_similarity final_rank_score -12.7062 -0.432939 10 3 Pose
Z57985071
[H]N(C(=O)C[C@H]1S/C(=N/c2ccccc2)N(CCc2cn([H])c3ccccc23)C1=O)c1ccccc1F
T09
native IFP available
T09
dockmulti_91311c650f2e_T09
0.854 1.000 0.583 native_similarity final_rank_score -26.6264 -0.713732 16 2 Pose
Z57985071
[H]N(C(=O)C[C@@H]1S/C(=N/c2ccccc2)N(CCc2cn([H])c3ccccc23)C1=O)c1ccccc1F
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.843 1.000 0.550 native_similarity final_rank_score -11.8896 -0.51517 15 3 Pose
Z57985071
[H]N(C(=O)C[C@@H]1S/C(=N/c2ccccc2)N(CCc2cn([H])c3ccccc23)C1=O)c1ccccc1F
T03
native IFP available
T03
dockmulti_91311c650f2e_T03
0.820 1.000 0.486 native_similarity final_rank_score -16.1408 -0.729107 18 1 Pose
Z57985071
[H]N(C(=O)C[C@H]1S/C(=N/c2ccccc2)N(CCc2cn([H])c3ccccc23)C1=O)c1ccccc1F
T02
native IFP available
T02
dockmulti_91311c650f2e_T02
0.798 1.000 0.424 native_similarity final_rank_score -22.1906 -0.658548 18 0 Pose
Z57985071
[H]N(C(=O)C[C@H]1S/C(=N/c2ccccc2)N(CCc2cn([H])c3ccccc23)C1=O)c1ccccc1F
T18
native IFP available
T18
dockmulti_91311c650f2e_T18
0.785 1.000 0.385 native_similarity final_rank_score -16.2628 -0.482362 11 1 Pose