FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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3 compounds in matrix 5 best compound-target hits listed 5 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T03T14T15T16T20
Z56958950
[H]N(C(=O)CN1C(=O)/C(=C2\SC(=S)N([C@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccc(OC)cc1
0.953 0.953 1 0.95
Z56958950
[H]N(C(=O)CN1C(=O)/C(=C2\SC(=S)N([C@@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccc(OC)cc1
0.883 0.820 3 0.88 0.83 0.75
Z56958950
[H]N(C(=O)CN1C(=O)/C(=C2/SC(=S)N([C@@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccc(OC)cc1
0.797 0.797 1 0.80

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z56958950
[H]N(C(=O)CN1C(=O)/C(=C2\SC(=S)N([C@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccc(OC)cc1
T20
native IFP available
T20
dockmulti_91311c650f2e_T20
0.953 1.000 0.867 native_similarity final_rank_score -16.5887 -0.468497 12 4 Pose
Z56958950
[H]N(C(=O)CN1C(=O)/C(=C2\SC(=S)N([C@@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccc(OC)cc1
T03
native IFP available
T03
dockmulti_91311c650f2e_T03
0.883 1.000 0.665 native_similarity final_rank_score -20.8548 -0.688871 19 2 Pose
Z56958950
[H]N(C(=O)CN1C(=O)/C(=C2\SC(=S)N([C@@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccc(OC)cc1
T15
native IFP available
T15
dockmulti_91311c650f2e_T15
0.829 1.000 0.513 native_similarity final_rank_score -18.8535 -0.580927 15 4 Pose
Z56958950
[H]N(C(=O)CN1C(=O)/C(=C2/SC(=S)N([C@@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccc(OC)cc1
T14
native IFP available
T14
dockmulti_91311c650f2e_T14
0.797 1.000 0.420 native_similarity final_rank_score -17.7419 -0.480056 14 3 Pose
Z56958950
[H]N(C(=O)CN1C(=O)/C(=C2\SC(=S)N([C@@H]3CCS(=O)(=O)C3)C2=O)c2ccccc21)c1ccc(OC)cc1
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.749 1.000 0.283 native_similarity final_rank_score -20.8405 -0.568762 12 1 Pose