FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
Reset
2 compounds in matrix 12 best compound-target hits listed 12 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T03T04T06T07T08T11T12T14T18T20T21
Z56821211
[H]Oc1cc(/C=N\N([H])C(=O)CSc2nc3ccccc3n2C)ccc1O
0.932 0.849 6 0.93 0.79 0.89 0.81 0.81 0.87
Z56821211
[H]Oc1ccc(/C=N/N([H])C(=O)CSc2nc3ccccc3n2C)cc1O
0.855 0.812 6 0.83 0.81 0.76 0.85 0.82 0.79

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z56821211
[H]Oc1cc(/C=N\N([H])C(=O)CSc2nc3ccccc3n2C)ccc1O
T06
native IFP available
T06
dockmulti_91311c650f2e_T06
0.932 1.000 0.807 native_similarity final_rank_score -21.1051 -0.887602 18 8 Pose
Z56821211
[H]Oc1cc(/C=N\N([H])C(=O)CSc2nc3ccccc3n2C)ccc1O
T11
native IFP available
T11
dockmulti_91311c650f2e_T11
0.890 0.952 0.773 native_similarity final_rank_score -23.3759 -1.01448 16 5 Pose
Z56821211
[H]Oc1cc(/C=N\N([H])C(=O)CSc2nc3ccccc3n2C)ccc1O
T21
native IFP available
T21
dockmulti_91311c650f2e_T21
0.867 1.000 0.621 native_similarity final_rank_score -23.2077 -0.880396 14 8 Pose
Z56821211
[H]Oc1ccc(/C=N/N([H])C(=O)CSc2nc3ccccc3n2C)cc1O
T07
native IFP available
T07
dockmulti_91311c650f2e_T07
0.855 1.000 0.585 native_similarity final_rank_score -27.9972 -1.20566 14 7 Pose
Z56821211
[H]Oc1ccc(/C=N/N([H])C(=O)CSc2nc3ccccc3n2C)cc1O
T02
native IFP available
T02
dockmulti_91311c650f2e_T02
0.832 1.000 0.519 native_similarity final_rank_score -20.5534 -0.90782 17 2 Pose
Z56821211
[H]Oc1ccc(/C=N/N([H])C(=O)CSc2nc3ccccc3n2C)cc1O
T14
native IFP available
T14
dockmulti_91311c650f2e_T14
0.821 1.000 0.489 native_similarity final_rank_score -15.628 -0.744972 13 8 Pose
Z56821211
[H]Oc1cc(/C=N\N([H])C(=O)CSc2nc3ccccc3n2C)ccc1O
T12
native IFP available
T12
dockmulti_91311c650f2e_T12
0.814 1.000 0.469 native_similarity final_rank_score -22.6426 -0.886933 16 7 Pose
Z56821211
[H]Oc1ccc(/C=N/N([H])C(=O)CSc2nc3ccccc3n2C)cc1O
T03
native IFP available
T03
dockmulti_91311c650f2e_T03
0.813 1.000 0.465 native_similarity final_rank_score -22.4888 -1.02375 16 4 Pose
Z56821211
[H]Oc1cc(/C=N\N([H])C(=O)CSc2nc3ccccc3n2C)ccc1O
T20
native IFP available
T20
dockmulti_91311c650f2e_T20
0.805 1.000 0.443 native_similarity final_rank_score -17.6431 -0.730464 9 6 Pose
Z56821211
[H]Oc1ccc(/C=N/N([H])C(=O)CSc2nc3ccccc3n2C)cc1O
T18
native IFP available
T18
dockmulti_91311c650f2e_T18
0.789 1.000 0.397 native_similarity final_rank_score -16.1327 -0.698745 15 7 Pose
Z56821211
[H]Oc1cc(/C=N\N([H])C(=O)CSc2nc3ccccc3n2C)ccc1O
T08
native IFP available
T08
dockmulti_91311c650f2e_T08
0.785 1.000 0.386 native_similarity final_rank_score -32.2234 -1.22625 12 6 Pose
Z56821211
[H]Oc1ccc(/C=N/N([H])C(=O)CSc2nc3ccccc3n2C)cc1O
T04
native IFP available
T04
dockmulti_91311c650f2e_T04
0.763 1.000 0.322 native_similarity final_rank_score -21.1412 -0.830943 10 0 Pose