FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
Reset
2 compounds in matrix 5 best compound-target hits listed 5 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T07T09T11T14T20
Z49558975
[H]Oc1ccc(/C=N\N([H])C(=O)c2ccc3c(c2)nc(C)n3CC)c(O[H])c1O[H]
0.894 0.820 4 0.89 0.82 0.77 0.80
Z49558975
[H]Oc1ccc(/C=N/N([H])C(=O)c2ccc3c(c2)[n+]([H])c(C)n3CC)c(O[H])c1O[H]
0.873 0.873 1 0.87

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z49558975
[H]Oc1ccc(/C=N\N([H])C(=O)c2ccc3c(c2)nc(C)n3CC)c(O[H])c1O[H]
T07
native IFP available
T07
dockmulti_91311c650f2e_T07
0.894 1.000 0.696 native_similarity final_rank_score -25.3441 -1.11963 14 8 Pose
Z49558975
[H]Oc1ccc(/C=N/N([H])C(=O)c2ccc3c(c2)[n+]([H])c(C)n3CC)c(O[H])c1O[H]
T11
native IFP available
T11
dockmulti_91311c650f2e_T11
0.873 1.000 0.638 native_similarity final_rank_score -24.6432 -0.951518 18 7 Pose
Z49558975
[H]Oc1ccc(/C=N\N([H])C(=O)c2ccc3c(c2)nc(C)n3CC)c(O[H])c1O[H]
T09
native IFP available
T09
dockmulti_91311c650f2e_T09
0.820 1.000 0.487 native_similarity final_rank_score -17.9625 -0.851112 16 4 Pose
Z49558975
[H]Oc1ccc(/C=N\N([H])C(=O)c2ccc3c(c2)nc(C)n3CC)c(O[H])c1O[H]
T20
native IFP available
T20
dockmulti_91311c650f2e_T20
0.799 1.000 0.425 native_similarity final_rank_score -20.1413 -0.799809 10 6 Pose
Z49558975
[H]Oc1ccc(/C=N\N([H])C(=O)c2ccc3c(c2)nc(C)n3CC)c(O[H])c1O[H]
T14
native IFP available
T14
dockmulti_91311c650f2e_T14
0.769 1.000 0.340 native_similarity final_rank_score -16.5296 -0.819026 12 7 Pose