FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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2 compounds in matrix 2 best compound-target hits listed 2 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T03T17
Z48204477
[H]n1c(C)c(C(=O)/C(C#N)=c2/s/c(=C\c3ccncc3)c(=O)n2-c2c(C)cccc2C)c2ccccc21
0.892 0.892 1 0.89
Z48204477
[H]n1c(C)c(C(=O)/C(C#N)=c2\s/c(=C/c3cc[n+]([H])cc3)c(=O)n2-c2c(C)cccc2C)c2ccccc21
0.807 0.807 1 0.81

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z48204477
[H]n1c(C)c(C(=O)/C(C#N)=c2/s/c(=C\c3ccncc3)c(=O)n2-c2c(C)cccc2C)c2ccccc21
T03
native IFP available
T03
selection_import_t03
0.892 1.000 0.690 native_similarity final_rank_score -21.9238 -0.753463 18 1 Pose
Z48204477
[H]n1c(C)c(C(=O)/C(C#N)=c2\s/c(=C/c3cc[n+]([H])cc3)c(=O)n2-c2c(C)cccc2C)c2ccccc21
T17
native IFP available
T17
selection_import_t17
0.807 1.000 0.450 native_similarity final_rank_score -20.5424 -0.626966 18 1 Pose