FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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4 compounds in matrix 7 best compound-target hits listed 7 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T03T09T11T14T15T16
Z2786555116
[H]N(C(=O)c1cccnc1)[C@H](c1ccc(OC)cc1)c1cc(Cl)c2ccc[n+]([H])c2c1O
0.900 0.826 3 0.82 0.90 0.76
Z2786555116
[H]N(C(=O)c1cccnc1)[C@@H](c1ccc(OC)cc1)c1cc(Cl)c2ccc[n+]([H])c2c1O
0.856 0.856 1 0.86
Z2786555116
[H]Oc1c([C@H](c2ccc(OC)cc2)N([H])C(=O)c2cccnc2)cc(Cl)c2cccnc12
0.810 0.810 1 0.81
Z2786555116
[H]Oc1c([C@@H](c2ccc(OC)cc2)N([H])C(=O)c2cccnc2)cc(Cl)c2cccnc12
0.786 0.761 2 0.74 0.79

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z2786555116
[H]N(C(=O)c1cccnc1)[C@H](c1ccc(OC)cc1)c1cc(Cl)c2ccc[n+]([H])c2c1O
T03
native IFP available
T03
dockmulti_91311c650f2e_T03
0.900 1.000 0.715 native_similarity final_rank_score -26.6523 -0.954123 17 3 Pose
Z2786555116
[H]N(C(=O)c1cccnc1)[C@@H](c1ccc(OC)cc1)c1cc(Cl)c2ccc[n+]([H])c2c1O
T09
native IFP available
T09
dockmulti_91311c650f2e_T09
0.856 1.000 0.589 native_similarity final_rank_score -21.6178 -0.782173 19 4 Pose
Z2786555116
[H]N(C(=O)c1cccnc1)[C@H](c1ccc(OC)cc1)c1cc(Cl)c2ccc[n+]([H])c2c1O
T02
native IFP available
T02
dockmulti_91311c650f2e_T02
0.823 1.000 0.493 native_similarity final_rank_score -19.513 -0.682302 17 2 Pose
Z2786555116
[H]Oc1c([C@H](c2ccc(OC)cc2)N([H])C(=O)c2cccnc2)cc(Cl)c2cccnc12
T14
native IFP available
T14
dockmulti_91311c650f2e_T14
0.810 1.000 0.458 native_similarity final_rank_score -21.8026 -0.752651 11 4 Pose
Z2786555116
[H]Oc1c([C@@H](c2ccc(OC)cc2)N([H])C(=O)c2cccnc2)cc(Cl)c2cccnc12
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.786 1.000 0.388 native_similarity final_rank_score -20.4819 -0.692178 13 5 Pose
Z2786555116
[H]N(C(=O)c1cccnc1)[C@H](c1ccc(OC)cc1)c1cc(Cl)c2ccc[n+]([H])c2c1O
T15
native IFP available
T15
dockmulti_91311c650f2e_T15
0.756 1.000 0.302 native_similarity final_rank_score -20.5324 -0.707757 14 6 Pose
Z2786555116
[H]Oc1c([C@@H](c2ccc(OC)cc2)N([H])C(=O)c2cccnc2)cc(Cl)c2cccnc12
T11
native IFP available
T11
dockmulti_91311c650f2e_T11
0.737 1.000 0.248 native_similarity final_rank_score -18.059 -0.670581 18 2 Pose