FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
Reset
2 compounds in matrix 5 best compound-target hits listed 5 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T05T09T14T20
Z226978722
[H][n+]1c(CSc2nc3ccccc3c3nc(C)nn23)cn2ccccc21
0.881 0.842 3 0.88 0.86 0.78
Z226978722
Cc1nc2c3ccccc3nc(SCc3cn4ccccc4n3)n2n1
0.834 0.832 2 0.83 0.83

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z226978722
[H][n+]1c(CSc2nc3ccccc3c3nc(C)nn23)cn2ccccc21
T02
native IFP available
T02
selection_import_t02
0.881 1.000 0.660 native_similarity final_rank_score -25.4511 -1.05712 18 1 Pose
Z226978722
[H][n+]1c(CSc2nc3ccccc3c3nc(C)nn23)cn2ccccc21
T09
native IFP available
T09
selection_import_t09
0.861 1.000 0.602 native_similarity final_rank_score -25.606 -1.01505 18 1 Pose
Z226978722
Cc1nc2c3ccccc3nc(SCc3cn4ccccc4n3)n2n1
T20
native IFP available
T20
selection_import_t20
0.834 1.000 0.525 native_similarity final_rank_score -19.1614 -0.77488 6 4 Pose
Z226978722
Cc1nc2c3ccccc3nc(SCc3cn4ccccc4n3)n2n1
T05
native IFP available
T05
selection_import_t05
0.830 1.000 0.514 native_similarity final_rank_score -26.0407 -1.1234 12 4 Pose
Z226978722
[H][n+]1c(CSc2nc3ccccc3c3nc(C)nn23)cn2ccccc21
T14
native IFP available
T14
selection_import_t14
0.783 1.000 0.380 native_similarity final_rank_score -23.9573 -0.984052 13 6 Pose