FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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2 compounds in matrix 4 best compound-target hits listed 4 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T03T08T21
Z19222909
[H]n1c(C)c(C(=O)[C@H](C)Sc2nnc(-c3ccccc3)c(-c3ccccc3)n2)c2ccccc21
0.890 0.864 2 0.84 0.89
Z19222909
[H]n1c(C)c(C(=O)[C@@H](C)Sc2nnc(-c3ccccc3)c(-c3ccccc3)n2)c2ccccc21
0.881 0.871 2 0.88 0.86

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z19222909
[H]n1c(C)c(C(=O)[C@H](C)Sc2nnc(-c3ccccc3)c(-c3ccccc3)n2)c2ccccc21
T21
native IFP available
T21
dockmulti_91311c650f2e_T21
0.890 1.000 0.686 native_similarity final_rank_score -24.2512 -0.836071 19 8 Pose
Z19222909
[H]n1c(C)c(C(=O)[C@@H](C)Sc2nnc(-c3ccccc3)c(-c3ccccc3)n2)c2ccccc21
T02
native IFP available
T02
dockmulti_91311c650f2e_T02
0.881 1.000 0.660 native_similarity final_rank_score -28.609 -0.912299 18 1 Pose
Z19222909
[H]n1c(C)c(C(=O)[C@@H](C)Sc2nnc(-c3ccccc3)c(-c3ccccc3)n2)c2ccccc21
T03
native IFP available
T03
dockmulti_91311c650f2e_T03
0.862 1.000 0.605 native_similarity final_rank_score -26.5051 -0.909874 17 1 Pose
Z19222909
[H]n1c(C)c(C(=O)[C@H](C)Sc2nnc(-c3ccccc3)c(-c3ccccc3)n2)c2ccccc21
T08
native IFP available
T08
dockmulti_91311c650f2e_T08
0.837 1.000 0.536 native_similarity final_rank_score -23.9638 -0.951389 17 3 Pose