FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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3 compounds in matrix 3 best compound-target hits listed 3 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T03T16
OSA_Lib_97
[H][N+]1([C@]23C[C@H](OC(=O)c4cccnc4)[C@H]([C@@H](c4ccccc4)C2)[C@@H](c2ccccc2)C3)CCCCC1
0.866 0.866 1 0.87
OSA_Lib_97
[H][N+]1([C@]23C[C@H](OC(=O)c4cccnc4)[C@H]([C@@H](c4ccccc4)C2)[C@H](c2ccccc2)C3)CCCCC1
0.838 0.838 1 0.84
OSA_Lib_97
[H][N+]1([C@@]23C[C@H](OC(=O)c4cccnc4)[C@@H]([C@@H](c4ccccc4)C2)[C@H](c2ccccc2)C3)CCCCC1
0.782 0.782 1 0.78

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OSA_Lib_97
[H][N+]1([C@]23C[C@H](OC(=O)c4cccnc4)[C@H]([C@@H](c4ccccc4)C2)[C@@H](c2ccccc2)C3)CCCCC1
T02
native IFP available
T02
dockmulti_91311c650f2e_T02
0.866 1.000 0.617 native_similarity final_rank_score -12.8736 -0.695403 21 1 Pose
OSA_Lib_97
[H][N+]1([C@]23C[C@H](OC(=O)c4cccnc4)[C@H]([C@@H](c4ccccc4)C2)[C@H](c2ccccc2)C3)CCCCC1
T03
native IFP available
T03
dockmulti_91311c650f2e_T03
0.838 1.000 0.538 native_similarity final_rank_score -15.1941 -0.633768 21 1 Pose
OSA_Lib_97
[H][N+]1([C@@]23C[C@H](OC(=O)c4cccnc4)[C@@H]([C@@H](c4ccccc4)C2)[C@H](c2ccccc2)C3)CCCCC1
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.782 1.000 0.378 native_similarity final_rank_score -14.2098 -0.50486 14 1 Pose