FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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4 compounds in matrix 6 best compound-target hits listed 6 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T03T11T15T16T18
OSA_Lib_89
[H]N(C(=O)CN1CCN(C)CC1)[C@H]1C[C@]2([N+]([H])(C)C)C[C@@H](c3ccccc3)[C@H]1[C@H](c1ccccc1)C2
0.854 0.854 1 0.85
OSA_Lib_89
[H]N(C(=O)CN1CC[N+]([H])(C)CC1)[C@@H]1C[C@]2([N+]([H])(C)C)C[C@@H](c3ccccc3)[C@H]1[C@H](c1ccccc1)C2
0.850 0.850 1 0.85
OSA_Lib_89
[H]N(C(=O)C[N+]1([H])CCN(C)CC1)[C@@H]1C[C@]2([N+]([H])(C)C)C[C@H](c3ccccc3)[C@H]1[C@H](c1ccccc1)C2
0.843 0.833 2 0.84 0.82
OSA_Lib_89
[H]N(C(=O)C[N+]1([H])CCN(C)CC1)[C@@H]1C[C@@]2([N+]([H])(C)C)C[C@H](c3ccccc3)[C@@H]1[C@H](c1ccccc1)C2
0.841 0.811 2 0.84 0.78

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OSA_Lib_89
[H]N(C(=O)CN1CCN(C)CC1)[C@H]1C[C@]2([N+]([H])(C)C)C[C@@H](c3ccccc3)[C@H]1[C@H](c1ccccc1)C2
T03
native IFP available
T03
dockmulti_91311c650f2e_T03
0.854 0.967 0.643 native_similarity final_rank_score -31.1721 -0.913339 21 1 Pose
OSA_Lib_89
[H]N(C(=O)CN1CC[N+]([H])(C)CC1)[C@@H]1C[C@]2([N+]([H])(C)C)C[C@@H](c3ccccc3)[C@H]1[C@H](c1ccccc1)C2
T11
native IFP available
T11
dockmulti_91311c650f2e_T11
0.850 1.000 0.570 native_similarity final_rank_score -17.9314 -0.456922 14 2 Pose
OSA_Lib_89
[H]N(C(=O)C[N+]1([H])CCN(C)CC1)[C@@H]1C[C@]2([N+]([H])(C)C)C[C@H](c3ccccc3)[C@H]1[C@H](c1ccccc1)C2
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.843 1.000 0.550 native_similarity final_rank_score -21.682 -0.574529 15 2 Pose
OSA_Lib_89
[H]N(C(=O)C[N+]1([H])CCN(C)CC1)[C@@H]1C[C@@]2([N+]([H])(C)C)C[C@H](c3ccccc3)[C@@H]1[C@H](c1ccccc1)C2
T02
native IFP available
T02
dockmulti_91311c650f2e_T02
0.841 0.986 0.570 native_similarity final_rank_score -22.4917 -0.673671 20 0 Pose
OSA_Lib_89
[H]N(C(=O)C[N+]1([H])CCN(C)CC1)[C@@H]1C[C@]2([N+]([H])(C)C)C[C@H](c3ccccc3)[C@H]1[C@H](c1ccccc1)C2
T18
native IFP available
T18
dockmulti_91311c650f2e_T18
0.823 0.988 0.516 native_similarity final_rank_score -21.7302 -0.518624 11 1 Pose
OSA_Lib_89
[H]N(C(=O)C[N+]1([H])CCN(C)CC1)[C@@H]1C[C@@]2([N+]([H])(C)C)C[C@H](c3ccccc3)[C@@H]1[C@H](c1ccccc1)C2
T15
native IFP available
T15
dockmulti_91311c650f2e_T15
0.780 1.000 0.373 native_similarity final_rank_score -13.0368 -0.440533 12 2 Pose