FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
Reset
2 compounds in matrix 4 best compound-target hits listed 4 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T02T09T16
OSA_Lib_314
[H][N+]1([C@]23C[C@H](c4ccccc4)[C@H](CN(C(=O)CN4C=CC(N5CCCC5)=CC4(C)C)C2)[C@H](c2ccccc2)C3)CCCC1
0.850 0.820 3 0.84 0.85 0.77
OSA_Lib_314
[H][N+]1([C@@]23C[C@H](c4ccccc4)[C@@H](CN(C(=O)CN4C=CC(N5CCCC5)=CC4(C)C)C2)[C@H](c2ccccc2)C3)CCCC1
0.795 0.795 1 0.80

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OSA_Lib_314
[H][N+]1([C@]23C[C@H](c4ccccc4)[C@H](CN(C(=O)CN4C=CC(N5CCCC5)=CC4(C)C)C2)[C@H](c2ccccc2)C3)CCCC1
T02
native IFP available
T02
selection_import_t02
0.850 1.000 0.570 native_similarity final_rank_score -23.8436 -0.625621 20 0 Pose
OSA_Lib_314
[H][N+]1([C@]23C[C@H](c4ccccc4)[C@H](CN(C(=O)CN4C=CC(N5CCCC5)=CC4(C)C)C2)[C@H](c2ccccc2)C3)CCCC1
T01
native IFP available
T01
selection_import_t01
0.838 1.000 0.539 native_similarity final_rank_score -24.5038 -0.627082 19 0 Pose
OSA_Lib_314
[H][N+]1([C@@]23C[C@H](c4ccccc4)[C@@H](CN(C(=O)CN4C=CC(N5CCCC5)=CC4(C)C)C2)[C@H](c2ccccc2)C3)CCCC1
T09
native IFP available
T09
selection_import_t09
0.795 1.000 0.415 native_similarity final_rank_score -23.5758 -0.620625 19 1 Pose
OSA_Lib_314
[H][N+]1([C@]23C[C@H](c4ccccc4)[C@H](CN(C(=O)CN4C=CC(N5CCCC5)=CC4(C)C)C2)[C@H](c2ccccc2)C3)CCCC1
T16
native IFP available
T16
selection_import_t16
0.773 1.000 0.352 native_similarity final_rank_score -21.3162 -0.543888 17 1 Pose