FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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2 compounds in matrix 5 best compound-target hits listed 5 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T08T09T15T16
OSA_Lib_304
[H]N1C[C@H]2[C@@H](c3ccccc3)C[C@]([N@+]([H])(C)Cc3ccccn3)(C[C@H]2c2ccccc2)C1
0.861 0.802 4 0.86 0.79 0.78 0.77
OSA_Lib_304
[H]N1C[C@H]2[C@H](c3ccccc3)C[C@]([N@+]([H])(C)Cc3ccccn3)(C[C@H]2c2ccccc2)C1
0.819 0.819 1 0.82

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OSA_Lib_304
[H]N1C[C@H]2[C@@H](c3ccccc3)C[C@]([N@+]([H])(C)Cc3ccccn3)(C[C@H]2c2ccccc2)C1
T02
native IFP available
T02
dockmulti_91311c650f2e_T02
0.861 0.992 0.617 native_similarity final_rank_score -23.7392 -0.759734 20 0 Pose
OSA_Lib_304
[H]N1C[C@H]2[C@H](c3ccccc3)C[C@]([N@+]([H])(C)Cc3ccccn3)(C[C@H]2c2ccccc2)C1
T09
native IFP available
T09
dockmulti_91311c650f2e_T09
0.819 0.991 0.500 native_similarity final_rank_score -19.5439 -0.702808 15 1 Pose
OSA_Lib_304
[H]N1C[C@H]2[C@@H](c3ccccc3)C[C@]([N@+]([H])(C)Cc3ccccn3)(C[C@H]2c2ccccc2)C1
T08
native IFP available
T08
dockmulti_91311c650f2e_T08
0.793 1.000 0.408 native_similarity final_rank_score -20.231 -0.642742 12 1 Pose
OSA_Lib_304
[H]N1C[C@H]2[C@@H](c3ccccc3)C[C@]([N@+]([H])(C)Cc3ccccn3)(C[C@H]2c2ccccc2)C1
T15
native IFP available
T15
dockmulti_91311c650f2e_T15
0.784 0.992 0.397 native_similarity final_rank_score -19.154 -0.644587 15 2 Pose
OSA_Lib_304
[H]N1C[C@H]2[C@@H](c3ccccc3)C[C@]([N@+]([H])(C)Cc3ccccn3)(C[C@H]2c2ccccc2)C1
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.769 0.960 0.414 native_similarity final_rank_score -17.4925 -0.659438 16 1 Pose