FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
Reset
2 compounds in matrix 4 best compound-target hits listed 4 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T09T15T16
OSA_Lib_278
[H]N1C[C@H]2[C@H](c3ccccc3)C[C@]([N@+]([H])(C)CCCC[N+]3([H])CCCC3)(C[C@H]2c2ccccc2)C1
0.829 0.799 3 0.81 0.83 0.76
OSA_Lib_278
[H]N1C[C@H]2[C@H](c3ccccc3)C[C@](N(C)CCCC[N+]3([H])CCCC3)(C[C@H]2c2ccccc2)C1
0.788 0.788 1 0.79

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OSA_Lib_278
[H]N1C[C@H]2[C@H](c3ccccc3)C[C@]([N@+]([H])(C)CCCC[N+]3([H])CCCC3)(C[C@H]2c2ccccc2)C1
T15
native IFP available
T15
dockmulti_91311c650f2e_T15
0.829 1.000 0.513 native_similarity final_rank_score -18.5849 -0.60833 15 0 Pose
OSA_Lib_278
[H]N1C[C@H]2[C@H](c3ccccc3)C[C@]([N@+]([H])(C)CCCC[N+]3([H])CCCC3)(C[C@H]2c2ccccc2)C1
T09
native IFP available
T09
dockmulti_91311c650f2e_T09
0.805 1.000 0.444 native_similarity final_rank_score -16.0956 -0.599022 17 2 Pose
OSA_Lib_278
[H]N1C[C@H]2[C@H](c3ccccc3)C[C@](N(C)CCCC[N+]3([H])CCCC3)(C[C@H]2c2ccccc2)C1
T02
native IFP available
T02
dockmulti_91311c650f2e_T02
0.788 1.000 0.394 native_similarity final_rank_score -17.6772 -0.634253 17 0 Pose
OSA_Lib_278
[H]N1C[C@H]2[C@H](c3ccccc3)C[C@]([N@+]([H])(C)CCCC[N+]3([H])CCCC3)(C[C@H]2c2ccccc2)C1
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.763 1.000 0.322 native_similarity final_rank_score -22.2008 -0.694319 14 3 Pose