FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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5 compounds in matrix 5 best compound-target hits listed 5 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T03T15T16T18
OSA_Lib_241
[H][N+]1(CCC[N@@+]2([H])CC[C@]3([N+]4([H])CCCCC4)C[C@@H](c4ccccc4)[C@H]2[C@H](c2ccccc2)C3)CCCCC1
0.838 0.838 1 0.84
OSA_Lib_241
[H][N+]1(CCC[N@@+]2([H])CC[C@@]3([N+]4([H])CCCCC4)C[C@H](c4ccccc4)[C@@H]2[C@H](c2ccccc2)C3)CCCCC1
0.834 0.834 1 0.83
OSA_Lib_241
[H][N+]1(CCC[N@@+]2([H])CC[C@]3([N+]4([H])CCCCC4)C[C@H](c4ccccc4)[C@H]2[C@@H](c2ccccc2)C3)CCCCC1
0.824 0.824 1 0.82
OSA_Lib_241
[H][N+]1(CCC[N@@+]2([H])CC[C@]3([N+]4([H])CCCCC4)C[C@H](c4ccccc4)[C@H]2[C@H](c2ccccc2)C3)CCCCC1
0.821 0.821 1 0.82
OSA_Lib_241
[H][N+]1(CCC[N@+]2([H])CC[C@]3(N4CCCCC4)C[C@H](c4ccccc4)[C@H]2[C@@H](c2ccccc2)C3)CCCCC1
0.818 0.818 1 0.82

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OSA_Lib_241
[H][N+]1(CCC[N@@+]2([H])CC[C@]3([N+]4([H])CCCCC4)C[C@@H](c4ccccc4)[C@H]2[C@H](c2ccccc2)C3)CCCCC1
T03
native IFP available
T03
dockmulti_91311c650f2e_T03
0.838 1.000 0.538 native_similarity final_rank_score -25.3389 -0.698908 21 1 Pose
OSA_Lib_241
[H][N+]1(CCC[N@@+]2([H])CC[C@@]3([N+]4([H])CCCCC4)C[C@H](c4ccccc4)[C@@H]2[C@H](c2ccccc2)C3)CCCCC1
T02
native IFP available
T02
dockmulti_91311c650f2e_T02
0.834 1.000 0.526 native_similarity final_rank_score -17.7004 -0.633841 20 0 Pose
OSA_Lib_241
[H][N+]1(CCC[N@@+]2([H])CC[C@]3([N+]4([H])CCCCC4)C[C@H](c4ccccc4)[C@H]2[C@@H](c2ccccc2)C3)CCCCC1
T18
native IFP available
T18
dockmulti_91311c650f2e_T18
0.824 1.000 0.497 native_similarity final_rank_score -13.2098 -0.413389 12 1 Pose
OSA_Lib_241
[H][N+]1(CCC[N@@+]2([H])CC[C@]3([N+]4([H])CCCCC4)C[C@H](c4ccccc4)[C@H]2[C@H](c2ccccc2)C3)CCCCC1
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.821 0.976 0.534 native_similarity final_rank_score -12.2708 -0.530567 16 1 Pose
OSA_Lib_241
[H][N+]1(CCC[N@+]2([H])CC[C@]3(N4CCCCC4)C[C@H](c4ccccc4)[C@H]2[C@@H](c2ccccc2)C3)CCCCC1
T15
native IFP available
T15
dockmulti_91311c650f2e_T15
0.818 0.989 0.498 native_similarity final_rank_score -13.9418 -0.490743 16 1 Pose