FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
Reset
2 compounds in matrix 3 best compound-target hits listed 3 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T15T16
OSA_Lib_199
[H][N+]1([C@]23C[C@H](c4ccccc4)[C@H]([C@@H](c4ccccc4)C2)[C@H](OC(=O)/C=C/c2ccccc2)C3)CCCCC1
0.846 0.841 2 0.85 0.84
OSA_Lib_199
[H][N+]1([C@]23C[C@H](OC(=O)/C=C/c4ccccc4)[C@H]([C@H](c4ccccc4)C2)[C@H](c2ccccc2)C3)CCCCC1
0.809 0.809 1 0.81

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OSA_Lib_199
[H][N+]1([C@]23C[C@H](c4ccccc4)[C@H]([C@@H](c4ccccc4)C2)[C@H](OC(=O)/C=C/c2ccccc2)C3)CCCCC1
T15
native IFP available
T15
dockmulti_91311c650f2e_T15
0.846 1.000 0.559 native_similarity final_rank_score -23.6634 -0.609681 16 0 Pose
OSA_Lib_199
[H][N+]1([C@]23C[C@H](c4ccccc4)[C@H]([C@@H](c4ccccc4)C2)[C@H](OC(=O)/C=C/c2ccccc2)C3)CCCCC1
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.837 1.000 0.534 native_similarity final_rank_score -19.6537 -0.558622 16 0 Pose
OSA_Lib_199
[H][N+]1([C@]23C[C@H](OC(=O)/C=C/c4ccccc4)[C@H]([C@H](c4ccccc4)C2)[C@H](c2ccccc2)C3)CCCCC1
T02
native IFP available
T02
dockmulti_91311c650f2e_T02
0.809 0.961 0.526 native_similarity final_rank_score -14.8885 -0.584676 20 0 Pose