FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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3 compounds in matrix 4 best compound-target hits listed 4 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T03T15T16T20
OSA_Lib_182
[H]N(CCC[N+]1([H])CCCC1)[C@H]1C[C@@]2([N+]3([H])CCN(C)CC3)C[C@H](c3ccccc3)[C@@H]1[C@H](c1ccccc1)C2
0.936 0.892 2 0.85 0.94
OSA_Lib_182
[H]N(CCC[N+]1([H])CCCC1)[C@@H]1C[C@]2([N+]3([H])CCN(C)CC3)C[C@H](c3ccccc3)[C@H]1[C@H](c1ccccc1)C2
0.904 0.904 1 0.90
OSA_Lib_182
[H][N+]1(C)CCN([C@]23C[C@H](c4ccccc4)[C@H]([C@H]([N+]([H])([H])CCC[N+]4([H])CCCC4)C2)[C@H](c2ccccc2)C3)CC1
0.810 0.810 1 0.81

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OSA_Lib_182
[H]N(CCC[N+]1([H])CCCC1)[C@H]1C[C@@]2([N+]3([H])CCN(C)CC3)C[C@H](c3ccccc3)[C@@H]1[C@H](c1ccccc1)C2
T20
native IFP available
T20
dockmulti_91311c650f2e_T20
0.936 1.000 0.817 native_similarity final_rank_score -13.4807 -0.359237 10 2 Pose
OSA_Lib_182
[H]N(CCC[N+]1([H])CCCC1)[C@@H]1C[C@]2([N+]3([H])CCN(C)CC3)C[C@H](c3ccccc3)[C@H]1[C@H](c1ccccc1)C2
T03
native IFP available
T03
dockmulti_91311c650f2e_T03
0.904 0.982 0.760 native_similarity final_rank_score -17.9378 -0.62423 20 1 Pose
OSA_Lib_182
[H]N(CCC[N+]1([H])CCCC1)[C@H]1C[C@@]2([N+]3([H])CCN(C)CC3)C[C@H](c3ccccc3)[C@@H]1[C@H](c1ccccc1)C2
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.848 0.991 0.582 native_similarity final_rank_score -16.7321 -0.513447 17 4 Pose
OSA_Lib_182
[H][N+]1(C)CCN([C@]23C[C@H](c4ccccc4)[C@H]([C@H]([N+]([H])([H])CCC[N+]4([H])CCCC4)C2)[C@H](c2ccccc2)C3)CC1
T15
native IFP available
T15
dockmulti_91311c650f2e_T15
0.810 0.961 0.530 native_similarity final_rank_score -20.2225 -0.562988 18 0 Pose