FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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4 compounds in matrix 4 best compound-target hits listed 4 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T15T16T18T20
OSA_Lib_181
[H][N+]1(CCC[N+]([H])([H])[C@@H]2C[C@]3([N+]4([H])CCCCC4)C[C@@H](c4ccccc4)[C@H]2[C@H](c2ccccc2)C3)CCCC1
0.917 0.917 1 0.92
OSA_Lib_181
[H][N+]1(CCC[N+]([H])([H])[C@H]2C[C@@]3([N+]4([H])CCCCC4)C[C@H](c4ccccc4)[C@@H]2[C@H](c2ccccc2)C3)CCCC1
0.838 0.838 1 0.84
OSA_Lib_181
[H][N+]1(CCC[N+]([H])([H])[C@H]2C[C@]3([N+]4([H])CCCCC4)C[C@@H](c4ccccc4)[C@H]2[C@H](c2ccccc2)C3)CCCC1
0.820 0.820 1 0.82
OSA_Lib_181
[H][N+]1(CCC[N+]([H])([H])[C@H]2C[C@]3([N+]4([H])CCCCC4)C[C@H](c4ccccc4)[C@H]2[C@@H](c2ccccc2)C3)CCCC1
0.804 0.804 1 0.80

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OSA_Lib_181
[H][N+]1(CCC[N+]([H])([H])[C@@H]2C[C@]3([N+]4([H])CCCCC4)C[C@@H](c4ccccc4)[C@H]2[C@H](c2ccccc2)C3)CCCC1
T20
native IFP available
T20
dockmulti_91311c650f2e_T20
0.917 1.000 0.763 native_similarity final_rank_score -12.6574 -0.51171 13 3 Pose
OSA_Lib_181
[H][N+]1(CCC[N+]([H])([H])[C@H]2C[C@@]3([N+]4([H])CCCCC4)C[C@H](c4ccccc4)[C@@H]2[C@H](c2ccccc2)C3)CCCC1
T18
native IFP available
T18
dockmulti_91311c650f2e_T18
0.838 1.000 0.538 native_similarity final_rank_score -15.0138 -0.470713 10 2 Pose
OSA_Lib_181
[H][N+]1(CCC[N+]([H])([H])[C@H]2C[C@]3([N+]4([H])CCCCC4)C[C@@H](c4ccccc4)[C@H]2[C@H](c2ccccc2)C3)CCCC1
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.820 1.000 0.485 native_similarity final_rank_score -14.2026 -0.525948 15 1 Pose
OSA_Lib_181
[H][N+]1(CCC[N+]([H])([H])[C@H]2C[C@]3([N+]4([H])CCCCC4)C[C@H](c4ccccc4)[C@H]2[C@@H](c2ccccc2)C3)CCCC1
T15
native IFP available
T15
dockmulti_91311c650f2e_T15
0.804 1.000 0.441 native_similarity final_rank_score -23.7163 -0.705885 16 3 Pose