FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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2 compounds in matrix 3 best compound-target hits listed 3 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T11T18T21
OHD_TB2022_10
[H]N([H])c1c2cc(OC)c(OC)cc2nc(N2CCN(C(=O)Cc3cccc(OC)c3)CC2)[n+]1[H]
0.907 0.871 2 0.91 0.84
OHD_TB2022_10
[H]N([H])c1nc(N2CCN(C(=O)Cc3cccc(OC)c3)CC2)nc2cc(OC)c(OC)cc12
0.809 0.809 1 0.81

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OHD_TB2022_10
[H]N([H])c1c2cc(OC)c(OC)cc2nc(N2CCN(C(=O)Cc3cccc(OC)c3)CC2)[n+]1[H]
T11
native IFP available
T11
selection_import_t11
0.907 1.000 0.734 native_similarity final_rank_score -25.5471 -0.74586 17 6 Pose
OHD_TB2022_10
[H]N([H])c1c2cc(OC)c(OC)cc2nc(N2CCN(C(=O)Cc3cccc(OC)c3)CC2)[n+]1[H]
T21
native IFP available
T21
selection_import_t21
0.835 1.000 0.529 native_similarity final_rank_score -24.5295 -0.748769 15 6 Pose
OHD_TB2022_10
[H]N([H])c1nc(N2CCN(C(=O)Cc3cccc(OC)c3)CC2)nc2cc(OC)c(OC)cc12
T18
native IFP available
T18
selection_import_t18
0.809 1.000 0.453 native_similarity final_rank_score -22.8622 -0.710288 15 3 Pose