FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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2 compounds in matrix 3 best compound-target hits listed 3 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T03T09T22
OHD_TB2020_9
[H]N(C(=O)c1cccc2c1N([H])C(C)(C)C[C@H]2C)[C@H](/C=C/S(=O)(=O)c1ccccc1)CCc1ccccc1
0.857 0.857 1 0.86
OHD_TB2020_9
[H]N(C(=O)c1cccc2c1[N+]([H])([H])C(C)(C)C[C@H]2C)[C@H](/C=C/S(=O)(=O)c1ccccc1)CCc1ccccc1
0.838 0.815 2 0.79 0.84

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OHD_TB2020_9
[H]N(C(=O)c1cccc2c1N([H])C(C)(C)C[C@H]2C)[C@H](/C=C/S(=O)(=O)c1ccccc1)CCc1ccccc1
T03
native IFP available
T03
selection_import_t03
0.857 1.000 0.591 native_similarity final_rank_score -27.4766 -0.829035 18 2 Pose
OHD_TB2020_9
[H]N(C(=O)c1cccc2c1[N+]([H])([H])C(C)(C)C[C@H]2C)[C@H](/C=C/S(=O)(=O)c1ccccc1)CCc1ccccc1
T22
native IFP available
T22
selection_import_t22
0.838 1.000 0.538 native_similarity final_rank_score -30.8531 -0.992946 22 6 Pose
OHD_TB2020_9
[H]N(C(=O)c1cccc2c1[N+]([H])([H])C(C)(C)C[C@H]2C)[C@H](/C=C/S(=O)(=O)c1ccccc1)CCc1ccccc1
T09
native IFP available
T09
selection_import_t09
0.792 1.000 0.406 native_similarity final_rank_score -27.8619 -0.76965 17 3 Pose