FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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6 compounds in matrix 8 best compound-target hits listed 8 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T06T07T08T09T12T13T19T21
OHD_Leishmania_93
[H]O[C@H]1[C@H]2c3cc4c(cc3C[N@@+]3([H])CCC(=C[C@H]1O[H])[C@@H]23)OCO4
0.894 0.830 3 0.82 0.78 0.89
OHD_Leishmania_93
[H]O[C@@H]1[C@@H]2c3cc4c(cc3C[N@+]3([H])CCC(=C[C@@H]1O[H])[C@@H]23)OCO4
0.876 0.876 1 0.88
OHD_Leishmania_93
[H]O[C@@H]1[C@H]2c3cc4c(cc3C[N@+]3([H])CCC(=C[C@H]1O[H])[C@@H]23)OCO4
0.838 0.838 1 0.84
OHD_Leishmania_93
[H]O[C@H]1[C@@H]2c3cc4c(cc3C[N@@+]3([H])CCC(=C[C@H]1O[H])[C@H]23)OCO4
0.826 0.826 1 0.83
OHD_Leishmania_93
[H]O[C@@H]1[C@@H]2c3cc4c(cc3CN3CCC(=C[C@H]1O[H])[C@H]23)OCO4
0.800 0.800 1 0.80
OHD_Leishmania_93
[H]O[C@H]1[C@H]2c3cc4c(cc3CN3CCC(=C[C@@H]1O[H])[C@H]23)OCO4
0.737 0.737 1 0.74

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OHD_Leishmania_93
[H]O[C@H]1[C@H]2c3cc4c(cc3C[N@@+]3([H])CCC(=C[C@H]1O[H])[C@@H]23)OCO4
T21
native IFP available
T21
dockmulti_91311c650f2e_T21
0.894 1.000 0.696 native_similarity final_rank_score -18.4534 -0.885439 14 7 Pose
OHD_Leishmania_93
[H]O[C@@H]1[C@@H]2c3cc4c(cc3C[N@+]3([H])CCC(=C[C@@H]1O[H])[C@@H]23)OCO4
T06
native IFP available
T06
dockmulti_91311c650f2e_T06
0.876 0.997 0.652 native_similarity final_rank_score -21.0114 -1.07315 18 4 Pose
OHD_Leishmania_93
[H]O[C@@H]1[C@H]2c3cc4c(cc3C[N@+]3([H])CCC(=C[C@H]1O[H])[C@@H]23)OCO4
T09
native IFP available
T09
dockmulti_91311c650f2e_T09
0.838 1.000 0.537 native_similarity final_rank_score -19.4042 -0.900635 16 1 Pose
OHD_Leishmania_93
[H]O[C@H]1[C@@H]2c3cc4c(cc3C[N@@+]3([H])CCC(=C[C@H]1O[H])[C@H]23)OCO4
T08
native IFP available
T08
dockmulti_91311c650f2e_T08
0.826 1.000 0.502 native_similarity final_rank_score -23.9637 -1.11875 12 2 Pose
OHD_Leishmania_93
[H]O[C@H]1[C@H]2c3cc4c(cc3C[N@@+]3([H])CCC(=C[C@H]1O[H])[C@@H]23)OCO4
T07
native IFP available
T07
dockmulti_91311c650f2e_T07
0.818 1.000 0.479 native_similarity final_rank_score -25.5475 -1.20663 13 1 Pose
OHD_Leishmania_93
[H]O[C@@H]1[C@@H]2c3cc4c(cc3CN3CCC(=C[C@H]1O[H])[C@H]23)OCO4
T12
native IFP available
T12
dockmulti_91311c650f2e_T12
0.800 1.000 0.428 native_similarity final_rank_score -22.8627 -1.08779 13 4 Pose
OHD_Leishmania_93
[H]O[C@H]1[C@H]2c3cc4c(cc3C[N@@+]3([H])CCC(=C[C@H]1O[H])[C@@H]23)OCO4
T13
native IFP available
T13
dockmulti_91311c650f2e_T13
0.778 1.000 0.364 native_similarity final_rank_score -17.0018 -0.793874 10 4 Pose
OHD_Leishmania_93
[H]O[C@H]1[C@H]2c3cc4c(cc3CN3CCC(=C[C@@H]1O[H])[C@H]23)OCO4
T19
native IFP available
T19
dockmulti_91311c650f2e_T19
0.737 0.979 0.288 native_similarity final_rank_score -26.9835 -1.26641 15 5 Pose