FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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2 compounds in matrix 4 best compound-target hits listed 4 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T03T07T08T09
OHD_Leishmania_131
[H]N([H])c1nc(N([H])[H])c2nc(CN(C)c3ccc(C(=O)N4CCCCC4)cc3)cnc2n1
0.953 0.938 3 0.94 0.92 0.95
OHD_Leishmania_131
[H]N([H])c1nc(N([H])[H])c2c(ncc(CN(C)c3ccc(C(=O)N4CCCCC4)cc3)[n+]2[H])n1
0.924 0.924 1 0.92

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OHD_Leishmania_131
[H]N([H])c1nc(N([H])[H])c2nc(CN(C)c3ccc(C(=O)N4CCCCC4)cc3)cnc2n1
T09
native IFP available
T09
dockmulti_91311c650f2e_T09
0.953 1.000 0.867 native_similarity final_rank_score -22.7525 -0.791827 20 10 Pose
OHD_Leishmania_131
[H]N([H])c1nc(N([H])[H])c2nc(CN(C)c3ccc(C(=O)N4CCCCC4)cc3)cnc2n1
T03
native IFP available
T03
dockmulti_91311c650f2e_T03
0.943 1.000 0.837 native_similarity final_rank_score -23.6866 -0.889546 20 10 Pose
OHD_Leishmania_131
[H]N([H])c1nc(N([H])[H])c2c(ncc(CN(C)c3ccc(C(=O)N4CCCCC4)cc3)[n+]2[H])n1
T07
native IFP available
T07
dockmulti_91311c650f2e_T07
0.924 1.000 0.784 native_similarity final_rank_score -39.6445 -1.32585 19 7 Pose
OHD_Leishmania_131
[H]N([H])c1nc(N([H])[H])c2nc(CN(C)c3ccc(C(=O)N4CCCCC4)cc3)cnc2n1
T08
native IFP available
T08
dockmulti_91311c650f2e_T08
0.917 1.000 0.763 native_similarity final_rank_score -37.6645 -1.23023 17 7 Pose