FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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2 compounds in matrix 4 best compound-target hits listed 4 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T03T09T16
OHD_ACDS_32
[H]N(CC(C)C)CC(c1cn([H])c2cc(Br)ccc12)c1cn([H])c2cc(Br)ccc12
0.916 0.895 2 0.92 0.87
OHD_ACDS_32
[H]n1cc(C(C[N+]([H])([H])CC(C)C)c2cn([H])c3cc(Br)ccc23)c2ccc(Br)cc21
0.872 0.854 2 0.87 0.84

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OHD_ACDS_32
[H]N(CC(C)C)CC(c1cn([H])c2cc(Br)ccc12)c1cn([H])c2cc(Br)ccc12
T02
native IFP available
T02
dockmulti_91311c650f2e_T02
0.916 1.000 0.760 native_similarity final_rank_score -20.5691 -0.918738 21 3 Pose
OHD_ACDS_32
[H]N(CC(C)C)CC(c1cn([H])c2cc(Br)ccc12)c1cn([H])c2cc(Br)ccc12
T03
native IFP available
T03
dockmulti_91311c650f2e_T03
0.874 1.000 0.639 native_similarity final_rank_score -20.0 -0.916949 18 3 Pose
OHD_ACDS_32
[H]n1cc(C(C[N+]([H])([H])CC(C)C)c2cn([H])c3cc(Br)ccc23)c2ccc(Br)cc21
T09
native IFP available
T09
dockmulti_91311c650f2e_T09
0.872 1.000 0.634 native_similarity final_rank_score -24.7735 -0.961296 19 2 Pose
OHD_ACDS_32
[H]n1cc(C(C[N+]([H])([H])CC(C)C)c2cn([H])c3cc(Br)ccc23)c2ccc(Br)cc21
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.837 1.000 0.534 native_similarity final_rank_score -15.7367 -0.786435 16 3 Pose