FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
Reset
1 compounds in matrix 15 best compound-target hits listed 15 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T02T04T05T06T08T09T11T12T14T15T17T18T21T22
NMT-TY0601
[H]N([H])c1c(NS(=O)(=O)c2ccc(N([H])C(C)=O)cc2)c(=O)nc(SCc2ccccc2)n1[H]
0.931 0.834 15 0.84 0.78 0.83 0.84 0.86 0.87 0.77 0.87 0.92 0.80 0.80 0.79 0.81 0.93 0.80

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
NMT-TY0601
[H]N([H])c1c(NS(=O)(=O)c2ccc(N([H])C(C)=O)cc2)c(=O)nc(SCc2ccccc2)n1[H]
T21
native IFP available
T21
selection_import_t21
0.931 1.000 0.803 native_similarity final_rank_score -25.47 -0.860345 17 12 Pose
NMT-TY0601
[H]N([H])c1c(NS(=O)(=O)c2ccc(N([H])C(C)=O)cc2)c(=O)nc(SCc2ccccc2)n1[H]
T12
native IFP available
T12
selection_import_t12
0.924 1.000 0.784 native_similarity final_rank_score -25.4028 -1.00124 16 9 Pose
NMT-TY0601
[H]N([H])c1c(NS(=O)(=O)c2ccc(N([H])C(C)=O)cc2)c(=O)nc(SCc2ccccc2)n1[H]
T11
native IFP available
T11
selection_import_t11
0.873 1.000 0.638 native_similarity final_rank_score -22.2524 -0.888004 13 5 Pose
NMT-TY0601
[H]N([H])c1c(NS(=O)(=O)c2ccc(N([H])C(C)=O)cc2)c(=O)nc(SCc2ccccc2)n1[H]
T08
native IFP available
T08
selection_import_t08
0.870 1.000 0.628 native_similarity final_rank_score -34.7998 -1.14564 16 11 Pose
NMT-TY0601
[H]N([H])c1c(NS(=O)(=O)c2ccc(N([H])C(C)=O)cc2)c(=O)nc(SCc2ccccc2)n1[H]
T06
native IFP available
T06
selection_import_t06
0.860 1.000 0.601 native_similarity final_rank_score -23.6414 -0.866114 20 3 Pose
NMT-TY0601
[H]N([H])c1c(NS(=O)(=O)c2ccc(N([H])C(C)=O)cc2)c(=O)nc(SCc2ccccc2)n1[H]
T05
native IFP available
T05
selection_import_t05
0.843 1.000 0.550 native_similarity final_rank_score -29.5939 -0.970487 15 10 Pose
NMT-TY0601
[H]N([H])c1c(NS(=O)(=O)c2ccc(N([H])C(C)=O)cc2)c(=O)nc(SCc2ccccc2)n1[H]
T01
native IFP available
T01
selection_import_t01
0.838 1.000 0.539 native_similarity final_rank_score -24.2954 -0.922656 19 3 Pose
NMT-TY0601
[H]N([H])c1c(NS(=O)(=O)c2ccc(N([H])C(C)=O)cc2)c(=O)nc(SCc2ccccc2)n1[H]
T04
native IFP available
T04
selection_import_t04
0.834 1.000 0.525 native_similarity final_rank_score -26.3515 -0.916521 14 1 Pose
NMT-TY0601
[H]N([H])c1c(NS(=O)(=O)c2ccc(N([H])C(C)=O)cc2)c(=O)nc(SCc2ccccc2)n1[H]
T18
native IFP available
T18
selection_import_t18
0.809 1.000 0.453 native_similarity final_rank_score -20.827 -0.754263 15 5 Pose
NMT-TY0601
[H]N([H])c1c(NS(=O)(=O)c2ccc(N([H])C(C)=O)cc2)c(=O)nc(SCc2ccccc2)n1[H]
T22
native IFP available
T22
selection_import_t22
0.804 1.000 0.440 native_similarity final_rank_score -33.9659 -1.11044 23 13 Pose
NMT-TY0601
[H]N([H])c1c(NS(=O)(=O)c2ccc(N([H])C(C)=O)cc2)c(=O)nc(SCc2ccccc2)n1[H]
T15
native IFP available
T15
selection_import_t15
0.797 1.000 0.421 native_similarity final_rank_score -21.0277 -0.803776 18 6 Pose
NMT-TY0601
[H]N([H])c1c(NS(=O)(=O)c2ccc(N([H])C(C)=O)cc2)c(=O)nc(SCc2ccccc2)n1[H]
T14
native IFP available
T14
selection_import_t14
0.797 1.000 0.420 native_similarity final_rank_score -23.4612 -0.780717 14 7 Pose
NMT-TY0601
[H]N([H])c1c(NS(=O)(=O)c2ccc(N([H])C(C)=O)cc2)c(=O)nc(SCc2ccccc2)n1[H]
T17
native IFP available
T17
selection_import_t17
0.786 1.000 0.389 native_similarity final_rank_score -23.7714 -0.846144 19 8 Pose
NMT-TY0601
[H]N([H])c1c(NS(=O)(=O)c2ccc(N([H])C(C)=O)cc2)c(=O)nc(SCc2ccccc2)n1[H]
T02
native IFP available
T02
selection_import_t02
0.777 1.000 0.363 native_similarity final_rank_score -24.8059 -0.8762 14 8 Pose
NMT-TY0601
[H]N([H])c1c(NS(=O)(=O)c2ccc(N([H])C(C)=O)cc2)c(=O)nc(SCc2ccccc2)n1[H]
T09
native IFP available
T09
selection_import_t09
0.771 1.000 0.347 native_similarity final_rank_score -30.8549 -0.984025 15 11 Pose