FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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2 compounds in matrix 6 best compound-target hits listed 6 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T03T06T08T13T19
KB_HAT_48
[H]N(C(=O)c1cnc(-c2cn([H])c3ncccc23)s1)[C@H](Cc1ccccc1)C[N+]([H])([H])[H]
0.890 0.838 3 0.89 0.82 0.81
KB_HAT_48
[H]N(C(=O)c1cnc(-c2cn([H])c3ncccc23)s1)[C@@H](Cc1ccccc1)C[N+]([H])([H])[H]
0.836 0.808 3 0.84 0.83 0.75

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
KB_HAT_48
[H]N(C(=O)c1cnc(-c2cn([H])c3ncccc23)s1)[C@H](Cc1ccccc1)C[N+]([H])([H])[H]
T02
native IFP available
T02
dockmulti_91311c650f2e_T02
0.890 1.000 0.687 native_similarity final_rank_score -23.7054 -1.02465 18 6 Pose
KB_HAT_48
[H]N(C(=O)c1cnc(-c2cn([H])c3ncccc23)s1)[C@@H](Cc1ccccc1)C[N+]([H])([H])[H]
T03
native IFP available
T03
dockmulti_91311c650f2e_T03
0.836 1.000 0.531 native_similarity final_rank_score -18.0037 -0.91976 18 1 Pose
KB_HAT_48
[H]N(C(=O)c1cnc(-c2cn([H])c3ncccc23)s1)[C@@H](Cc1ccccc1)C[N+]([H])([H])[H]
T13
native IFP available
T13
dockmulti_91311c650f2e_T13
0.835 1.000 0.527 native_similarity final_rank_score -21.37 -1.0614 16 8 Pose
KB_HAT_48
[H]N(C(=O)c1cnc(-c2cn([H])c3ncccc23)s1)[C@H](Cc1ccccc1)C[N+]([H])([H])[H]
T06
native IFP available
T06
dockmulti_91311c650f2e_T06
0.816 1.000 0.475 native_similarity final_rank_score -19.0266 -0.880775 17 1 Pose
KB_HAT_48
[H]N(C(=O)c1cnc(-c2cn([H])c3ncccc23)s1)[C@H](Cc1ccccc1)C[N+]([H])([H])[H]
T08
native IFP available
T08
dockmulti_91311c650f2e_T08
0.808 1.000 0.452 native_similarity final_rank_score -23.5798 -1.12947 14 3 Pose
KB_HAT_48
[H]N(C(=O)c1cnc(-c2cn([H])c3ncccc23)s1)[C@@H](Cc1ccccc1)C[N+]([H])([H])[H]
T19
native IFP available
T19
dockmulti_91311c650f2e_T19
0.752 1.000 0.293 native_similarity final_rank_score -25.5241 -1.21859 23 5 Pose