FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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2 compounds in matrix 6 best compound-target hits listed 6 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T03T09T16T18T20T21
KB_HAT_38
[H]O[C@H]1CC[N@+]([H])(Cc2cccc(-c3cccc(N([H])C(=O)c4ccc(C#N)cc4)c3)c2)CC1
0.897 0.821 3 0.81 0.76 0.90
KB_HAT_38
[H]OC1CCN(Cc2cccc(-c3cccc(N([H])C(=O)c4ccc(C#N)cc4)c3)c2)CC1
0.890 0.856 3 0.89 0.89 0.79

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
KB_HAT_38
[H]O[C@H]1CC[N@+]([H])(Cc2cccc(-c3cccc(N([H])C(=O)c4ccc(C#N)cc4)c3)c2)CC1
T21
native IFP available
T21
dockmulti_91311c650f2e_T21
0.897 1.000 0.706 native_similarity final_rank_score -23.1438 -0.755564 17 6 Pose
KB_HAT_38
[H]OC1CCN(Cc2cccc(-c3cccc(N([H])C(=O)c4ccc(C#N)cc4)c3)c2)CC1
T09
native IFP available
T09
dockmulti_91311c650f2e_T09
0.890 1.000 0.684 native_similarity final_rank_score -20.3634 -0.800245 19 3 Pose
KB_HAT_38
[H]OC1CCN(Cc2cccc(-c3cccc(N([H])C(=O)c4ccc(C#N)cc4)c3)c2)CC1
T03
native IFP available
T03
dockmulti_91311c650f2e_T03
0.886 1.000 0.673 native_similarity final_rank_score -24.162 -0.823752 19 1 Pose
KB_HAT_38
[H]O[C@H]1CC[N@+]([H])(Cc2cccc(-c3cccc(N([H])C(=O)c4ccc(C#N)cc4)c3)c2)CC1
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.807 1.000 0.450 native_similarity final_rank_score -20.4399 -0.697829 18 3 Pose
KB_HAT_38
[H]OC1CCN(Cc2cccc(-c3cccc(N([H])C(=O)c4ccc(C#N)cc4)c3)c2)CC1
T18
native IFP available
T18
dockmulti_91311c650f2e_T18
0.793 1.000 0.408 native_similarity final_rank_score -20.2303 -0.666846 14 2 Pose
KB_HAT_38
[H]O[C@H]1CC[N@+]([H])(Cc2cccc(-c3cccc(N([H])C(=O)c4ccc(C#N)cc4)c3)c2)CC1
T20
native IFP available
T20
dockmulti_91311c650f2e_T20
0.759 1.000 0.312 native_similarity final_rank_score -12.6009 -0.573698 13 3 Pose