FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
Reset
2 compounds in matrix 10 best compound-target hits listed 10 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T03T08T09T11T12T13T14T15T16T18
KB_HAT_172
[H]N(C(=O)C1CC1)[C@H]1CC[N@@+]([H])([C@@H]2Cc3ccc(NS(=O)(=O)c4cc(F)cc(F)c4)cc3C2)CC1
0.904 0.818 5 0.90 0.84 0.81 0.76 0.78
KB_HAT_172
[H]N(C(=O)C1CC1)[C@H]1CC[N@@+]([H])([C@H]2Cc3ccc(NS(=O)(=O)c4cc(F)cc(F)c4)cc3C2)CC1
0.864 0.812 5 0.80 0.86 0.84 0.79 0.76

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
KB_HAT_172
[H]N(C(=O)C1CC1)[C@H]1CC[N@@+]([H])([C@@H]2Cc3ccc(NS(=O)(=O)c4cc(F)cc(F)c4)cc3C2)CC1
T03
native IFP available
T03
dockmulti_91311c650f2e_T03
0.904 1.000 0.725 native_similarity final_rank_score -21.6745 -0.717074 19 2 Pose
KB_HAT_172
[H]N(C(=O)C1CC1)[C@H]1CC[N@@+]([H])([C@H]2Cc3ccc(NS(=O)(=O)c4cc(F)cc(F)c4)cc3C2)CC1
T12
native IFP available
T12
dockmulti_91311c650f2e_T12
0.864 1.000 0.613 native_similarity final_rank_score -12.7624 -0.568801 18 4 Pose
KB_HAT_172
[H]N(C(=O)C1CC1)[C@H]1CC[N@@+]([H])([C@H]2Cc3ccc(NS(=O)(=O)c4cc(F)cc(F)c4)cc3C2)CC1
T14
native IFP available
T14
dockmulti_91311c650f2e_T14
0.842 1.000 0.550 native_similarity final_rank_score -17.7677 -0.537158 17 3 Pose
KB_HAT_172
[H]N(C(=O)C1CC1)[C@H]1CC[N@@+]([H])([C@@H]2Cc3ccc(NS(=O)(=O)c4cc(F)cc(F)c4)cc3C2)CC1
T08
native IFP available
T08
dockmulti_91311c650f2e_T08
0.842 1.000 0.548 native_similarity final_rank_score -30.6016 -0.911223 16 3 Pose
KB_HAT_172
[H]N(C(=O)C1CC1)[C@H]1CC[N@@+]([H])([C@@H]2Cc3ccc(NS(=O)(=O)c4cc(F)cc(F)c4)cc3C2)CC1
T09
native IFP available
T09
dockmulti_91311c650f2e_T09
0.809 1.000 0.454 native_similarity final_rank_score -21.7454 -0.722711 19 2 Pose
KB_HAT_172
[H]N(C(=O)C1CC1)[C@H]1CC[N@@+]([H])([C@H]2Cc3ccc(NS(=O)(=O)c4cc(F)cc(F)c4)cc3C2)CC1
T11
native IFP available
T11
dockmulti_91311c650f2e_T11
0.802 1.000 0.433 native_similarity final_rank_score -16.8719 -0.638356 19 0 Pose
KB_HAT_172
[H]N(C(=O)C1CC1)[C@H]1CC[N@@+]([H])([C@H]2Cc3ccc(NS(=O)(=O)c4cc(F)cc(F)c4)cc3C2)CC1
T15
native IFP available
T15
dockmulti_91311c650f2e_T15
0.793 1.000 0.408 native_similarity final_rank_score -20.4523 -0.703616 14 5 Pose
KB_HAT_172
[H]N(C(=O)C1CC1)[C@H]1CC[N@@+]([H])([C@@H]2Cc3ccc(NS(=O)(=O)c4cc(F)cc(F)c4)cc3C2)CC1
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.779 1.000 0.368 native_similarity final_rank_score -17.3009 -0.571614 15 2 Pose
KB_HAT_172
[H]N(C(=O)C1CC1)[C@H]1CC[N@@+]([H])([C@H]2Cc3ccc(NS(=O)(=O)c4cc(F)cc(F)c4)cc3C2)CC1
T18
native IFP available
T18
dockmulti_91311c650f2e_T18
0.758 1.000 0.309 native_similarity final_rank_score -16.9306 -0.533284 13 2 Pose
KB_HAT_172
[H]N(C(=O)C1CC1)[C@H]1CC[N@@+]([H])([C@@H]2Cc3ccc(NS(=O)(=O)c4cc(F)cc(F)c4)cc3C2)CC1
T13
native IFP available
T13
dockmulti_91311c650f2e_T13
0.757 1.000 0.306 native_similarity final_rank_score -16.7595 -0.603964 18 2 Pose