FAIRMol

Z49724509

Pose ID 9750 Compound 1121 Pose 1171

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-1.004 kcal/mol/HA) ✓ Good fit quality (FQ -8.99) ✗ High strain energy (17.4 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-24.084
kcal/mol
LE
-1.004
kcal/mol/HA
Fit Quality
-8.99
FQ (Leeson)
HAC
24
heavy atoms
MW
409
Da
LogP
3.72
cLogP
Strain ΔE
17.4 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 17.4 kcal/mol

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 24 π–π 2 Clashes 9 Severe clashes 2
Final rank6.941663920851766Score-24.0835
Inter norm-0.956894Intra norm-0.067612
Top1000noExcludedyes
Contacts17H-bonds2
Artifact reasonexcluded; geometry warning; 8 clashes; 2 protein clashes; moderate strain Δ 19.7
ResiduesA:ALA34;A:ARG100;A:ARG59;A:GLN56;A:ILE160;A:ILE47;A:LEU90;A:LEU97;A:MET55;A:NDP301;A:PHE58;A:PHE94;A:PRO91;A:THR86;A:TYR166;A:VAL32;A:VAL33

Protein summary

223 residues
Protein targetT06Atoms3452
Residues223Chains1
Residue summaryARG:408; VAL:352; LYS:308; LEU:304; PRO:238; ILE:209; GLU:195; THR:182; SER:176; ALA:160; PHE:140; ASN:126; GLY:126; ASP:108; GLN:85; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name8RHTContacts21
PoseOpen native poseH-bonds6
IFP residuesA:ALA34; A:ASP54; A:HIS182; A:ILE160; A:ILE47; A:LEU90; A:LEU97; A:MET55; A:NDP301; A:PHE233; A:PHE58; A:PHE94; A:PRO91; A:SER89; A:THR184; A:THR86; A:TRP49; A:TYR166; A:TYR57; A:VAL32; A:VAL33
Current overlap14Native recall0.67
Jaccard0.58RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1207 2.430143154907441 -1.19382 -30.1867 6 15 0 0.00 0.00 - no Open
1201 2.4590174680979047 -1.26453 -31.8913 6 16 0 0.00 0.00 - no Open
1953 2.8400690927329624 -0.734472 -17.9639 5 9 0 0.00 0.00 - no Open
1908 3.305177520629858 -0.730958 -19.3589 5 12 0 0.00 0.00 - no Open
1958 3.6394876868458246 -0.763068 -17.911 6 10 0 0.00 0.00 - no Open
1955 3.6761661205884892 -0.55105 -11.9604 6 12 0 0.00 0.00 - no Open
1170 3.8348229988696003 -0.930798 -19.4897 0 17 15 0.71 0.00 - no Open
1563 4.5002173945509965 -1.1615 -23.9956 13 17 0 0.00 0.00 - no Open
1954 4.503117859188464 -0.728145 -16.7015 6 12 0 0.00 0.00 - no Open
1957 5.074169882563248 -0.815124 -17.3361 7 11 0 0.00 0.00 - yes Open
1567 5.4202018677778625 -0.888389 -15.7861 9 13 0 0.00 0.00 - yes Open
1565 5.4519267318111595 -1.45598 -31.2552 12 16 0 0.00 0.00 - yes Open
1956 5.751487436525558 -0.657139 -16.3227 5 9 0 0.00 0.00 - yes Open
1911 5.850036536798715 -0.950209 -26.6197 7 13 0 0.00 0.00 - yes Open
1172 6.386292556677911 -0.944628 -20.0632 1 17 14 0.67 0.00 - yes Open
1570 6.471207934876456 -1.05511 -25.0177 8 19 0 0.00 0.00 - yes Open
1568 6.531054243391047 -0.854058 -19.9371 6 17 0 0.00 0.00 - yes Open
1564 6.629182736230375 -1.15211 -25.1158 10 17 0 0.00 0.00 - yes Open
1168 6.664891527018511 -0.975766 -17.9682 1 17 14 0.67 0.00 - yes Open
1205 6.75309589925006 -1.18499 -32.4258 3 17 0 0.00 0.00 - yes Open
1171 6.941663920851766 -0.956894 -24.0835 2 17 14 0.67 0.00 - yes Current
1909 7.22878133022391 -0.920036 -23.2283 6 13 0 0.00 0.00 - yes Open
1569 7.248502876011524 -1.04523 -23.6535 9 15 0 0.00 0.00 - yes Open
1210 7.445536821069086 -1.11972 -27.0097 8 13 0 0.00 0.00 - yes Open
1910 7.878953770499661 -0.667251 -16.9474 7 14 0 0.00 0.00 - yes Open
1169 8.027539752005387 -0.990568 -25.18 3 16 13 0.62 0.00 - yes Open
1566 8.297213516026027 -1.06485 -24.7992 7 19 0 0.00 0.00 - yes Open
1204 8.390141378325266 -1.26016 -31.1285 9 13 0 0.00 0.00 - yes Open
1173 8.52512299003625 -0.761459 -19.3834 2 20 17 0.81 0.00 - yes Open
1202 10.037222800942548 -1.39302 -32.2253 6 19 0 0.00 0.00 - yes Open
1208 10.07271766611601 -1.23696 -30.1909 7 18 0 0.00 0.00 - yes Open
1209 10.204050037001787 -1.22425 -29.639 4 17 0 0.00 0.00 - yes Open
1206 10.367610776310922 -1.33226 -33.1999 7 18 0 0.00 0.00 - yes Open
1571 10.768799511203035 -1.08542 -22.8271 11 14 0 0.00 0.00 - yes Open
1572 11.085712337405427 -0.940268 -25.9868 8 16 0 0.00 0.00 - yes Open
1203 11.367536281309768 -1.31659 -30.4671 3 19 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -24.084kcal/mol
Ligand efficiency (LE) -1.0035kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -8.993
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 24HA

Physicochemical properties

Molecular weight 409.3Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.72
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 17.38kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 95.22kcal/mol
Minimised FF energy 77.84kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.