FAIRMol

Z108563960

Pose ID 9640 Compound 91 Pose 1061

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.770 kcal/mol/HA) ✓ Good fit quality (FQ -7.18) ✗ Very high strain energy (20.1 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-20.788
kcal/mol
LE
-0.770
kcal/mol/HA
Fit Quality
-7.18
FQ (Leeson)
HAC
27
heavy atoms
MW
377
Da
LogP
3.39
cLogP
Strain ΔE
20.1 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 20.1 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 3 Clashes 19 Severe clashes 0
Final rank8.435071689989822Score-20.788
Inter norm-0.858258Intra norm0.088331
Top1000noExcludedno
Contacts15H-bonds1
Artifact reasongeometry warning; 15 clashes; 19 protein contact clashes; moderate strain Δ 19.6
ResiduesA:ALA34;A:ARG59;A:ASP54;A:ILE47;A:LEU90;A:LEU97;A:MET55;A:NDP301;A:PHE58;A:PHE94;A:PRO91;A:THR184;A:TYR57;A:VAL32;A:VAL33

Protein summary

223 residues
Protein targetT06Atoms3452
Residues223Chains1
Residue summaryARG:408; VAL:352; LYS:308; LEU:304; PRO:238; ILE:209; GLU:195; THR:182; SER:176; ALA:160; PHE:140; ASN:126; GLY:126; ASP:108; GLN:85; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name8RHTContacts21
PoseOpen native poseH-bonds6
IFP residuesA:ALA34; A:ASP54; A:HIS182; A:ILE160; A:ILE47; A:LEU90; A:LEU97; A:MET55; A:NDP301; A:PHE233; A:PHE58; A:PHE94; A:PRO91; A:SER89; A:THR184; A:THR86; A:TRP49; A:TYR166; A:TYR57; A:VAL32; A:VAL33
Current overlap14Native recall0.67
Jaccard0.64RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1763 3.1886793116212595 -0.741479 -20.3801 2 10 0 0.00 0.00 - no Open
1762 3.3001366044298743 -0.728422 -20.2258 3 10 0 0.00 0.00 - no Open
2428 3.7138734046822024 -0.909823 -22.4282 1 17 1 0.05 0.00 - no Open
2460 3.746313313204172 -0.866501 -21.6002 1 14 0 0.00 0.00 - no Open
964 4.7098947576715355 -1.07448 -26.7837 2 16 0 0.00 0.00 - no Open
1061 8.435071689989822 -0.858258 -20.788 1 15 14 0.67 0.00 - no Current
965 5.31750172013611 -1.09833 -28.1058 3 16 0 0.00 0.00 - yes Open
2429 5.595893630632348 -0.97743 -23.6679 1 18 1 0.05 0.00 - yes Open
2459 6.595580972599691 -0.972905 -25.4432 2 17 0 0.00 0.00 - yes Open
1060 7.82507918816123 -0.873952 -22.2228 2 15 14 0.67 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -20.788kcal/mol
Ligand efficiency (LE) -0.7699kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.183
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 27HA

Physicochemical properties

Molecular weight 377.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.39
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 20.07kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 98.20kcal/mol
Minimised FF energy 78.13kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.