FAIRMol

KB_Leish_48

Pose ID 8968 Compound 1210 Pose 389

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.678 kcal/mol/HA) ✓ Good fit quality (FQ -6.24) ✗ High strain energy (17.7 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-17.620
kcal/mol
LE
-0.678
kcal/mol/HA
Fit Quality
-6.24
FQ (Leeson)
HAC
26
heavy atoms
MW
367
Da
LogP
3.69
cLogP
Strain ΔE
17.7 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 17.7 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 3 Clashes 15 Severe clashes 0
Final rank6.54930298271091Score-17.6196
Inter norm-0.861186Intra norm0.18351
Top1000noExcludedno
Contacts18H-bonds1
Artifact reasongeometry warning; 12 clashes; 15 protein contact clashes; moderate strain Δ 17.5
ResiduesA:ALA34;A:ARG59;A:ASP54;A:HIS182;A:ILE47;A:LEU90;A:LEU97;A:MET55;A:NDP301;A:PHE58;A:PHE94;A:PRO91;A:SER89;A:THR184;A:THR86;A:TYR57;A:VAL32;A:VAL33

Protein summary

223 residues
Protein targetT06Atoms3452
Residues223Chains1
Residue summaryARG:408; VAL:352; LYS:308; LEU:304; PRO:238; ILE:209; GLU:195; THR:182; SER:176; ALA:160; PHE:140; ASN:126; GLY:126; ASP:108; GLN:85; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name8RHTContacts21
PoseOpen native poseH-bonds6
IFP residuesA:ALA34; A:ASP54; A:HIS182; A:ILE160; A:ILE47; A:LEU90; A:LEU97; A:MET55; A:NDP301; A:PHE233; A:PHE58; A:PHE94; A:PRO91; A:SER89; A:THR184; A:THR86; A:TRP49; A:TYR166; A:TYR57; A:VAL32; A:VAL33
Current overlap17Native recall0.81
Jaccard0.77RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
514 3.9662958483665713 -1.01732 -26.0095 2 19 1 0.05 0.00 - no Open
520 4.301836178432678 -1.24956 -26.9896 8 15 0 0.00 0.00 - no Open
353 4.596450420236221 -1.07887 -32.1101 6 16 0 0.00 0.00 - no Open
672 4.753100092565043 -0.786201 -16.7503 5 10 0 0.00 0.00 - no Open
397 5.048193273144377 -1.04441 -18.5458 6 20 0 0.00 0.00 - no Open
387 5.840056262686303 -0.859948 -22.1403 0 19 17 0.81 0.00 - no Open
385 5.8674133039578855 -0.855196 -21.9631 1 19 17 0.81 0.00 - no Open
670 5.890359289671385 -0.61506 -16.5311 6 8 0 0.00 0.00 - no Open
389 6.54930298271091 -0.861186 -17.6196 1 18 17 0.81 0.00 - no Current
388 6.575484509827401 -0.861514 -17.4613 0 17 16 0.76 0.00 - no Open
386 7.031484444432119 -0.869502 -18.8868 0 18 16 0.76 0.00 - no Open
617 8.444381253918266 -0.945702 -19.3234 5 13 0 0.00 0.00 - no Open
515 5.002267750236572 -0.786048 -21.7552 2 18 1 0.05 0.00 - yes Open
671 5.675461707062585 -0.7826 -16.3145 5 10 0 0.00 0.00 - yes Open
521 6.259841322912159 -1.26883 -25.9434 11 16 0 0.00 0.00 - yes Open
669 6.297290514047962 -0.767859 -17.5137 4 9 0 0.00 0.00 - yes Open
616 7.085290123456148 -0.865828 -17.4641 6 12 0 0.00 0.00 - yes Open
355 8.935425138100962 -1.16958 -24.324 9 17 0 0.00 0.00 - yes Open
354 11.033255109762516 -0.996602 -26.325 8 14 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -17.620kcal/mol
Ligand efficiency (LE) -0.6777kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.244
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 26HA

Physicochemical properties

Molecular weight 366.8Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.69
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 17.70kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 41.22kcal/mol
Minimised FF energy 23.52kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.