FAIRMol

KB_HAT_10

Pose ID 8902 Compound 1164 Pose 323

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.690 kcal/mol/HA) ✓ Good fit quality (FQ -6.44) ✗ Very high strain energy (25.4 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-18.633
kcal/mol
LE
-0.690
kcal/mol/HA
Fit Quality
-6.44
FQ (Leeson)
HAC
27
heavy atoms
MW
387
Da
LogP
3.51
cLogP
Strain ΔE
25.4 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 25.4 kcal/mol

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 24 π–π 3 Clashes 7 Severe clashes 0
Final rank4.565915127752357Score-18.6325
Inter norm-0.856296Intra norm0.147579
Top1000noExcludedno
Contacts20H-bonds2
Artifact reasongeometry warning; 10 clashes; 7 protein contact clashes; high strain Δ 27.0
ResiduesA:ALA34;A:ARG100;A:ARG59;A:ASP54;A:HIS182;A:ILE160;A:ILE47;A:LEU90;A:LEU97;A:MET55;A:NDP301;A:PHE58;A:PHE94;A:PRO91;A:THR184;A:THR86;A:TYR166;A:TYR57;A:VAL32;A:VAL33

Protein summary

223 residues
Protein targetT06Atoms3452
Residues223Chains1
Residue summaryARG:408; VAL:352; LYS:308; LEU:304; PRO:238; ILE:209; GLU:195; THR:182; SER:176; ALA:160; PHE:140; ASN:126; GLY:126; ASP:108; GLN:85; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name8RHTContacts21
PoseOpen native poseH-bonds6
IFP residuesA:ALA34; A:ASP54; A:HIS182; A:ILE160; A:ILE47; A:LEU90; A:LEU97; A:MET55; A:NDP301; A:PHE233; A:PHE58; A:PHE94; A:PRO91; A:SER89; A:THR184; A:THR86; A:TRP49; A:TYR166; A:TYR57; A:VAL32; A:VAL33
Current overlap18Native recall0.86
Jaccard0.78RMSD-
H-bond strict1Strict recall0.20
H-bond same residue+role1Role recall0.25
H-bond same residue1Residue recall0.25

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
295 2.6248326995720337 -1.04839 -25.698 3 15 0 0.00 0.00 - no Open
419 3.895463271160683 -0.966028 -22.426 6 13 0 0.00 0.00 - no Open
323 4.565915127752357 -0.856296 -18.6325 2 20 18 0.86 0.25 - no Current
322 4.6996822258351765 -0.749027 -18.7433 3 18 17 0.81 0.25 - no Open
93 4.750220329559591 -1.01697 -20.9972 3 16 0 0.00 0.00 - no Open
319 4.787722288785993 -0.860322 -19.3331 2 20 18 0.86 0.25 - no Open
310 5.0017875109194385 -0.87165 -21.9792 4 17 0 0.00 0.00 - no Open
491 5.092797929141489 -0.869886 -18.9182 2 20 18 0.86 0.25 - no Open
87 5.431987139034222 -0.775495 -18.406 1 18 16 0.76 0.00 - no Open
106 5.495972486877 -0.809824 -21.3114 7 13 0 0.00 0.00 - no Open
490 5.5687415736876105 -0.776667 -17.7845 5 19 16 0.76 0.25 - no Open
454 5.606773355888093 -0.646318 -15.8114 7 11 0 0.00 0.00 - no Open
318 54.75142313912754 -0.773082 -18.2762 1 20 18 0.86 0.00 - no Open
453 6.415587053861709 -0.964684 -25.8709 8 13 0 0.00 0.00 - yes Open
88 54.780493194146516 -0.868266 -19.382 2 20 18 0.86 0.25 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -18.633kcal/mol
Ligand efficiency (LE) -0.6901kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.438
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 27HA

Physicochemical properties

Molecular weight 387.5Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.51
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 25.38kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 71.03kcal/mol
Minimised FF energy 45.65kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.