FAIRMol

OHD_TB2020_34

Pose ID 8790 Compound 5 Pose 211

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.791 kcal/mol/HA) ✓ Good fit quality (FQ -7.55) ✗ Very high strain energy (21.0 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-22.932
kcal/mol
LE
-0.791
kcal/mol/HA
Fit Quality
-7.55
FQ (Leeson)
HAC
29
heavy atoms
MW
432
Da
LogP
3.90
cLogP
Strain ΔE
21.0 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 21.0 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 4 Clashes 10 Severe clashes 0
Final rank4.874497153620346Score-22.932
Inter norm-0.89983Intra norm0.10907
Top1000noExcludedno
Contacts18H-bonds1
Artifact reasongeometry warning; 8 clashes; 10 protein contact clashes; high strain Δ 25.1
ResiduesA:ALA34;A:ARG100;A:ARG59;A:ASP54;A:GLN56;A:ILE160;A:ILE47;A:LEU90;A:LEU97;A:MET55;A:NDP301;A:PHE58;A:PHE94;A:PRO91;A:THR184;A:TYR57;A:VAL32;A:VAL33

Protein summary

223 residues
Protein targetT06Atoms3452
Residues223Chains1
Residue summaryARG:408; VAL:352; LYS:308; LEU:304; PRO:238; ILE:209; GLU:195; THR:182; SER:176; ALA:160; PHE:140; ASN:126; GLY:126; ASP:108; GLN:85; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name8RHTContacts21
PoseOpen native poseH-bonds6
IFP residuesA:ALA34; A:ASP54; A:HIS182; A:ILE160; A:ILE47; A:LEU90; A:LEU97; A:MET55; A:NDP301; A:PHE233; A:PHE58; A:PHE94; A:PRO91; A:SER89; A:THR184; A:THR86; A:TRP49; A:TYR166; A:TYR57; A:VAL32; A:VAL33
Current overlap15Native recall0.71
Jaccard0.62RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
229 1.9669914172748868 -0.765303 -21.6244 0 18 0 0.00 0.00 - no Open
228 3.5074251799698715 -0.892365 -25.6003 1 19 0 0.00 0.00 - no Open
211 4.874497153620346 -0.89983 -22.932 1 18 15 0.71 0.00 - no Current
210 5.771700032053993 -0.902347 -25.0526 1 16 14 0.67 0.00 - no Open
225 5.974682028343906 -0.646672 -17.8124 4 11 0 0.00 0.00 - no Open
102 6.2657967941064285 -0.947993 -25.7194 1 12 0 0.00 0.00 - no Open
101 6.001849678896553 -0.716527 -18.487 1 13 0 0.00 0.00 - yes Open
103 6.570221105490032 -0.855879 -22.7584 2 12 0 0.00 0.00 - yes Open
212 6.711389579232198 -0.801535 -21.6642 0 20 17 0.81 0.00 - yes Open
226 7.917648822636545 -0.633964 -16.612 5 9 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -22.932kcal/mol
Ligand efficiency (LE) -0.7908kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.548
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 29HA

Physicochemical properties

Molecular weight 432.3Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.90
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 21.01kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 48.93kcal/mol
Minimised FF energy 27.92kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.