FAIRMol

OHD_TB2020_31

Pose ID 8784 Compound 17 Pose 205

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.780 kcal/mol/HA) ✓ Good fit quality (FQ -7.53) ✗ Very high strain energy (20.8 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-23.412
kcal/mol
LE
-0.780
kcal/mol/HA
Fit Quality
-7.53
FQ (Leeson)
HAC
30
heavy atoms
MW
473
Da
LogP
4.79
cLogP
Strain ΔE
20.8 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 20.8 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 4 Clashes 14 Severe clashes 3
Final rank10.078743635315023Score-23.4118
Inter norm-0.827433Intra norm0.0470393
Top1000noExcludedyes
Contacts19H-bonds1
Artifact reasonexcluded; geometry warning; 9 clashes; 3 protein clashes; high strain Δ 27.2
ResiduesA:ALA34;A:ARG100;A:ARG59;A:ASP54;A:GLN56;A:ILE160;A:ILE47;A:LEU90;A:LEU97;A:MET55;A:NDP301;A:PHE58;A:PHE94;A:PRO91;A:THR184;A:TYR166;A:TYR57;A:VAL32;A:VAL33

Protein summary

223 residues
Protein targetT06Atoms3452
Residues223Chains1
Residue summaryARG:408; VAL:352; LYS:308; LEU:304; PRO:238; ILE:209; GLU:195; THR:182; SER:176; ALA:160; PHE:140; ASN:126; GLY:126; ASP:108; GLN:85; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name8RHTContacts21
PoseOpen native poseH-bonds6
IFP residuesA:ALA34; A:ASP54; A:HIS182; A:ILE160; A:ILE47; A:LEU90; A:LEU97; A:MET55; A:NDP301; A:PHE233; A:PHE58; A:PHE94; A:PRO91; A:SER89; A:THR184; A:THR86; A:TRP49; A:TYR166; A:TYR57; A:VAL32; A:VAL33
Current overlap16Native recall0.76
Jaccard0.67RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
227 2.590081390399253 -0.763217 -21.7991 1 20 0 0.00 0.00 - no Open
225 4.245710859034881 -0.841485 -25.5372 1 20 0 0.00 0.00 - no Open
206 5.658638579876223 -0.921707 -26.2863 0 16 14 0.67 0.00 - no Open
180 6.034110348717511 -1.01086 -30.362 6 15 0 0.00 0.00 - no Open
94 6.118311237264021 -0.66823 -19.3874 0 12 0 0.00 0.00 - no Open
226 6.481230590677507 -0.793212 -23.951 2 19 0 0.00 0.00 - yes Open
95 7.270870308065414 -0.940002 -28.3004 1 12 0 0.00 0.00 - yes Open
179 8.753531502642371 -1.08277 -30.7978 4 18 0 0.00 0.00 - yes Open
205 10.078743635315023 -0.827433 -23.4118 1 19 16 0.76 0.00 - yes Current
96 13.806205885947607 -0.841014 -22.9396 4 13 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -23.412kcal/mol
Ligand efficiency (LE) -0.7804kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.528
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 30HA

Physicochemical properties

Molecular weight 472.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 4.79
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 20.82kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 56.07kcal/mol
Minimised FF energy 35.25kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.