FAIRMol

OHD_Leishmania_93

Pose ID 8585 Compound 1043 Pose 6

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.873 kcal/mol/HA) ✓ Good fit quality (FQ -7.45) ✓ Good H-bonds (5 bonds) ✗ High strain energy (11.1 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-18.334
kcal/mol
LE
-0.873
kcal/mol/HA
Fit Quality
-7.45
FQ (Leeson)
HAC
21
heavy atoms
MW
288
Da
LogP
-0.67
cLogP
Strain ΔE
11.1 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 11.1 kcal/mol

Interaction summary

Collapsible panels
H-bonds 5 Hydrophobic 24 π–π 1 Clashes 9 Severe clashes 2
Final rank56.17914633995929Score-18.3336
Inter norm-0.870867Intra norm-0.00216024
Top1000noExcludedyes
Contacts18H-bonds5
Artifact reasonexcluded; geometry warning; 8 clashes; 2 protein clashes
ResiduesA:ALA34;A:ASP54;A:GLY161;A:ILE160;A:ILE47;A:LEU90;A:LEU97;A:MET55;A:NDP301;A:PHE58;A:PHE94;A:PRO91;A:THR184;A:THR86;A:TYR166;A:TYR57;A:VAL32;A:VAL33

Protein summary

223 residues
Protein targetT06Atoms3452
Residues223Chains1
Residue summaryARG:408; VAL:352; LYS:308; LEU:304; PRO:238; ILE:209; GLU:195; THR:182; SER:176; ALA:160; PHE:140; ASN:126; GLY:126; ASP:108; GLN:85; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name8RHTContacts21
PoseOpen native poseH-bonds6
IFP residuesA:ALA34; A:ASP54; A:HIS182; A:ILE160; A:ILE47; A:LEU90; A:LEU97; A:MET55; A:NDP301; A:PHE233; A:PHE58; A:PHE94; A:PRO91; A:SER89; A:THR184; A:THR86; A:TRP49; A:TYR166; A:TYR57; A:VAL32; A:VAL33
Current overlap17Native recall0.81
Jaccard0.77RMSD-
H-bond strict1Strict recall0.20
H-bond same residue+role1Role recall0.25
H-bond same residue3Residue recall0.75

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
22 1.8113138856378344 -0.957094 -20.1735 4 16 16 0.76 0.25 - no Open
46 1.8824936748035193 -0.949466 -20.032 3 16 16 0.76 0.25 - no Open
32 1.975897908401348 -1.07315 -21.0114 4 18 17 0.81 0.25 - no Open
35 2.3091522367316486 -0.967888 -20.5799 3 17 16 0.76 0.25 - no Open
41 2.720578612882062 -0.989048 -20.7352 2 16 16 0.76 0.25 - no Open
45 2.973615490461874 -0.984528 -20.7604 2 17 17 0.81 0.25 - no Open
28 51.97006187013032 -0.949752 -20.2992 3 18 18 0.86 0.25 - no Open
11 52.009940122072045 -1.00895 -21.7009 3 17 17 0.81 0.25 - no Open
13 52.235982438268486 -1.005 -21.1865 3 16 16 0.76 0.25 - no Open
36 52.25779620888597 -0.933889 -19.7422 3 18 17 0.81 0.25 - no Open
19 52.26671613765812 -0.981414 -20.9902 4 17 17 0.81 0.25 - no Open
14 52.306680314098514 -0.891535 -19.0899 4 17 17 0.81 0.25 - no Open
12 52.31325420681044 -0.860349 -18.2317 3 17 17 0.81 0.25 - no Open
30 52.51935565294619 -0.880989 -18.336 2 16 16 0.76 0.00 - no Open
27 52.60489882609083 -0.961728 -20.4673 2 16 16 0.76 0.25 - no Open
9 52.677095901860156 -0.824622 -17.6349 0 13 13 0.62 0.00 - no Open
21 52.71579714766378 -1.0058 -21.2287 3 17 17 0.81 0.25 - no Open
18 52.82285017495177 -0.903782 -19.0766 4 17 16 0.76 0.25 - no Open
37 52.844115628434835 -0.895373 -18.6878 4 17 17 0.81 0.25 - no Open
10 53.03240129688975 -0.882688 -18.6791 3 17 17 0.81 0.25 - no Open
38 53.312908271044066 -0.925106 -19.8252 4 18 17 0.81 0.25 - no Open
39 53.919151864140055 -0.912323 -19.3361 2 14 14 0.67 0.25 - no Open
51 54.45379486672558 -0.87523 -17.2609 3 18 17 0.81 0.25 - no Open
8 53.72648072346619 -0.954081 -19.6415 3 17 17 0.81 0.25 - yes Open
50 53.84105406752808 -0.868982 -18.0747 3 16 16 0.76 0.25 - yes Open
16 54.22778883483703 -0.91346 -19.5613 2 17 17 0.81 0.25 - yes Open
23 54.24398066113544 -0.983207 -20.7448 3 17 17 0.81 0.00 - yes Open
42 54.263431590298445 -0.929342 -19.7849 3 19 17 0.81 0.25 - yes Open
20 54.496803175338826 -0.910244 -18.7773 4 18 16 0.76 0.25 - yes Open
53 54.50827876605101 -0.943777 -19.805 4 19 17 0.81 0.25 - yes Open
26 54.53260611340698 -0.755785 -15.8424 2 15 14 0.67 0.00 - yes Open
15 54.59294249568364 -0.900637 -19.4349 3 18 16 0.76 0.25 - yes Open
24 55.32163917707414 -1.04641 -21.5716 4 18 17 0.81 0.25 - yes Open
6 56.17914633995929 -0.870867 -18.3336 5 18 17 0.81 0.25 - yes Current
43 56.34102127447972 -0.964116 -20.2501 2 15 14 0.67 0.25 - yes Open
48 56.600868003060846 -0.815154 -17.3252 3 14 14 0.67 0.25 - yes Open
33 56.799208960519756 -0.83737 -17.7561 4 14 14 0.67 0.00 - yes Open
52 57.61016152693548 -0.895258 -18.8098 4 16 15 0.71 0.00 - yes Open
34 57.64363332178546 -0.923328 -19.3593 4 16 15 0.71 0.00 - yes Open
47 58.03437934304549 -1.04549 -21.7757 3 17 15 0.71 0.00 - yes Open
40 58.30746740727956 -1.04956 -21.3648 4 16 14 0.67 0.00 - yes Open
17 58.312435633046775 -0.986089 -21.0373 5 15 14 0.67 0.25 - yes Open
25 58.414209805493186 -0.989075 -20.6398 3 17 15 0.71 0.00 - yes Open
44 58.71077859565911 -0.865488 -14.0748 4 15 14 0.67 0.00 - yes Open
29 59.12514025161087 -0.982772 -21.0374 2 17 15 0.71 0.00 - yes Open
31 59.294802684767006 -0.919968 -19.1283 5 14 14 0.67 0.25 - yes Open
49 59.30267829032168 -0.994632 -21.1268 2 17 15 0.71 0.00 - yes Open
7 60.12672878465521 -0.949923 -19.5461 3 17 15 0.71 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -18.334kcal/mol
Ligand efficiency (LE) -0.8730kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.447
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 21HA

Physicochemical properties

Molecular weight 288.3Da
Lipinski: ≤ 500 Da
LogP (cLogP) -0.67
Lipinski: ≤ 5
Rotatable bonds 0

Conformational strain (MMFF94s)

Strain energy (ΔE) 11.06kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 70.36kcal/mol
Minimised FF energy 59.30kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.