FAIRMol

Z45660418

Pose ID 8252 Compound 821 Pose 1665

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.925 kcal/mol/HA) ✓ Good fit quality (FQ -8.03) ✗ Very high strain energy (26.8 kcal/mol) ✗ No H-bonds detected ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-20.341
kcal/mol
LE
-0.925
kcal/mol/HA
Fit Quality
-8.03
FQ (Leeson)
HAC
22
heavy atoms
MW
359
Da
LogP
3.04
cLogP
Strain ΔE
26.8 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 26.8 kcal/mol

Interaction summary

Collapsible panels
H-bonds 0 Hydrophobic 23 π–π 3 Clashes 8 Severe clashes 0
Final rank4.097504252087317Score-20.3415
Inter norm-0.948423Intra norm0.0238093
Top1000noExcludedno
Contacts15H-bonds0
Artifact reasongeometry warning; 7 clashes; 8 protein contact clashes; high strain Δ 26.8
ResiduesA:ARG17;A:GLY225;A:HIS241;A:LEU188;A:LEU226;A:LEU229;A:MET233;A:NDP302;A:PHE113;A:SER111;A:SER227;A:TYR191;A:TYR194;A:VAL230;D:ARG287

Protein summary

308 residues
Protein targetT04Atoms4210
Residues308Chains3
Residue summaryLEU:494; ALA:421; ARG:384; VAL:368; THR:295; TYR:231; SER:198; PRO:196; ILE:190; LYS:176; ASN:154; GLU:150; GLY:126; PHE:120; HIS:119; ASP:108

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name7PXXContacts19
PoseOpen native poseH-bonds8
IFP residuesA:ARG17; A:ASP181; A:GLY225; A:HIS241; A:LEU188; A:LEU226; A:LEU229; A:LYS198; A:MET233; A:NDP302; A:PHE113; A:PRO115; A:SER111; A:SER112; A:SER227; A:TYR191; A:TYR194; A:VAL230; D:ARG287
Current overlap15Native recall0.79
Jaccard0.79RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

No hydrogen bonds detected for this pose.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1666 2.8069001591562426 -0.998323 -21.9856 0 15 15 0.79 0.00 - no Open
1665 4.097504252087317 -0.948423 -20.3415 0 15 15 0.79 0.00 - no Current

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -20.341kcal/mol
Ligand efficiency (LE) -0.9246kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -8.027
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 22HA

Physicochemical properties

Molecular weight 358.9Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.04
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 26.82kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 123.07kcal/mol
Minimised FF energy 96.25kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.