FAIRMol

OHD_Leishmania_216

Pose ID 81 Compound 246 Pose 81

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.775 kcal/mol/HA) ✓ Good fit quality (FQ -7.76) ✗ Very high strain energy (70.8 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-26.356
kcal/mol
LE
-0.775
kcal/mol/HA
Fit Quality
-7.76
FQ (Leeson)
HAC
34
heavy atoms
MW
507
Da
LogP
0.02
cLogP
Strain ΔE
70.8 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 70.8 kcal/mol

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 24 π–π 2 Clashes 8 Severe clashes 1
Final rank8.590315552454543Score-26.3559
Inter norm-0.673211Intra norm-0.101962
Top1000noExcludedyes
Contacts20H-bonds2
Artifact reasonexcluded; geometry warning; 9 clashes; 1 protein clash; high strain Δ 68.1
ResiduesA:ALA10;A:ARG29;A:ASN65;A:ASP22;A:GLU31;A:GLY117;A:ILE61;A:ILE8;A:LEU23;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:PRO62;A:SER60;A:THR137;A:THR57;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap18Native recall0.86
Jaccard0.78RMSD-
H-bond strict1Strict recall0.20
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
77 4.99971184383414 -0.658954 -34.6381 3 17 14 0.67 0.20 - no Open
58 5.016140314611698 -0.542019 -25.7359 3 16 0 0.00 0.00 - no Open
59 5.282395323491784 -0.554775 -29.4083 10 21 0 0.00 0.00 - no Open
57 5.477316230496473 -0.537155 -28.9035 4 19 0 0.00 0.00 - no Open
74 5.501881399456847 -0.51903 -25.3767 9 20 0 0.00 0.00 - no Open
29 5.814897333168477 -0.55621 -32.7894 12 20 0 0.00 0.00 - no Open
77 5.850034945805316 -0.518839 -32.9854 10 17 0 0.00 0.00 - no Open
79 6.196031634632424 -0.606531 -40.7304 7 14 0 0.00 0.00 - no Open
24 6.928372348970923 -0.609538 -25.6289 6 19 0 0.00 0.00 - no Open
55 7.1242553175212056 -0.457122 -33.0222 5 15 0 0.00 0.00 - no Open
53 8.397776211096767 -0.496004 -29.1286 6 14 0 0.00 0.00 - no Open
56 53.54183780799225 -0.605762 -28.7111 3 17 0 0.00 0.00 - no Open
78 54.01245522782489 -0.507718 -42.294 9 16 0 0.00 0.00 - no Open
76 6.1671465332990785 -0.64426 -30.6218 3 19 17 0.81 0.20 - yes Open
56 6.784112011299907 -0.62398 -47.4596 7 20 0 0.00 0.00 - yes Open
27 7.642161286869958 -0.688729 -35.0146 10 17 0 0.00 0.00 - yes Open
81 8.590315552454543 -0.673211 -26.3559 2 20 18 0.86 0.20 - yes Current
75 53.794483519417305 -0.415498 -25.8107 7 16 0 0.00 0.00 - yes Open
76 54.66896572278946 -0.643719 -29.1109 7 19 0 0.00 0.00 - yes Open
26 55.14834615685666 -0.592317 -24.8612 5 18 0 0.00 0.00 - yes Open
52 55.72414189247244 -0.593982 -29.1166 6 12 0 0.00 0.00 - yes Open
60 55.86889612413243 -0.586657 -37.0021 2 19 0 0.00 0.00 - yes Open
31 55.95408612524393 -0.690631 -36.1449 5 18 0 0.00 0.00 - yes Open
72 56.0339639993994 -0.533069 -24.5792 6 12 0 0.00 0.00 - yes Open
57 56.17765444723122 -0.699249 -10.1847 5 16 0 0.00 0.00 - yes Open
61 56.230275676396516 -0.804264 -40.0676 6 21 0 0.00 0.00 - yes Open
30 56.386656380410415 -0.567137 -44.7365 7 18 0 0.00 0.00 - yes Open
28 56.74825662793501 -0.489736 -20.9965 5 17 0 0.00 0.00 - yes Open
75 56.89840367677394 -0.654774 -36.4978 2 17 13 0.62 0.00 - yes Open
55 57.08883509170568 -0.642571 -32.4534 11 16 0 0.00 0.00 - yes Open
54 57.157439981367204 -0.551002 -21.5545 6 14 0 0.00 0.00 - yes Open
73 57.19145027814992 -0.477567 -28.4514 8 21 0 0.00 0.00 - yes Open
51 57.20480849231251 -0.451295 -27.5527 6 15 0 0.00 0.00 - yes Open
50 57.51145846999063 -0.578399 -25.3493 10 15 0 0.00 0.00 - yes Open
25 57.54084931829345 -0.664237 -35.1056 9 17 0 0.00 0.00 - yes Open
79 57.86290195805525 -0.688882 -40.6352 3 22 18 0.86 0.40 - yes Open
80 58.479409468065214 -0.913784 -49.6127 5 20 13 0.62 0.40 - yes Open
74 58.521262348407696 -0.639443 -22.9901 3 19 12 0.57 0.20 - yes Open
54 58.81339553950522 -0.690846 -30.7609 8 20 0 0.00 0.00 - yes Open
78 60.63875406873109 -0.636268 -25.7447 7 18 11 0.52 0.20 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -26.356kcal/mol
Ligand efficiency (LE) -0.7752kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.756
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 34HA

Physicochemical properties

Molecular weight 507.5Da
Lipinski: ≤ 500 Da
LogP (cLogP) 0.02
Lipinski: ≤ 5
Rotatable bonds 9

Conformational strain (MMFF94s)

Strain energy (ΔE) 70.82kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 43.06kcal/mol
Minimised FF energy -27.76kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.