FAIRMol

Z56786752

Pose ID 7968 Compound 801 Pose 1381

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-1.136 kcal/mol/HA) ✓ Good fit quality (FQ -9.31) ✓ Strong H-bond network (6 bonds) ✗ High strain energy (12.9 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-21.581
kcal/mol
LE
-1.136
kcal/mol/HA
Fit Quality
-9.31
FQ (Leeson)
HAC
19
heavy atoms
MW
269
Da
LogP
-1.00
cLogP
Strain ΔE
12.9 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 6 Hydrophobic 15 π–π 2 Clashes 7 Severe clashes 0
Final rank2.446321432702807Score-21.5812
Inter norm-1.18618Intra norm0.0503307
Top1000noExcludedno
Contacts12H-bonds6
Artifact reasongeometry warning; 4 clashes; 7 protein contact clashes; moderate strain Δ 15.7
ResiduesA:ARG17;A:GLY225;A:HIS241;A:LEU188;A:LEU226;A:LEU229;A:NDP302;A:PHE113;A:SER111;A:SER227;A:TYR194;D:ARG287

Protein summary

308 residues
Protein targetT04Atoms4210
Residues308Chains3
Residue summaryLEU:494; ALA:421; ARG:384; VAL:368; THR:295; TYR:231; SER:198; PRO:196; ILE:190; LYS:176; ASN:154; GLU:150; GLY:126; PHE:120; HIS:119; ASP:108

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name7PXXContacts19
PoseOpen native poseH-bonds8
IFP residuesA:ARG17; A:ASP181; A:GLY225; A:HIS241; A:LEU188; A:LEU226; A:LEU229; A:LYS198; A:MET233; A:NDP302; A:PHE113; A:PRO115; A:SER111; A:SER112; A:SER227; A:TYR191; A:TYR194; A:VAL230; D:ARG287
Current overlap12Native recall0.63
Jaccard0.63RMSD-
H-bond strict4Strict recall0.67
H-bond same residue+role3Role recall0.60
H-bond same residue3Residue recall0.60

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1381 2.446321432702807 -1.18618 -21.5812 6 12 12 0.63 0.60 - no Current
1383 4.079423833494527 -1.37069 -28.7921 4 11 11 0.58 0.40 - yes Open
1382 5.989028515139474 -1.26065 -19.3205 6 10 10 0.53 0.60 - yes Open
1380 56.72659682460353 -1.2716 -25.5639 2 11 11 0.58 0.40 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -21.581kcal/mol
Ligand efficiency (LE) -1.1359kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -9.310
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 19HA

Physicochemical properties

Molecular weight 269.2Da
Lipinski: ≤ 500 Da
LogP (cLogP) -1.00
Lipinski: ≤ 5
Rotatable bonds 2

Conformational strain (MMFF94s)

Strain energy (ΔE) 12.94kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 50.50kcal/mol
Minimised FF energy 37.57kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.