FAIRMol

KB_Leish_188

Pose ID 733 Compound 250 Pose 733

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing
T02
Dihydrofolate reductase Homo sapiens
Ligand KB_Leish_188
PDB5SD8

3D complex viewer

Strict H-bonds Permissive H-bonds
Viewer legend
Protein receptor
Pocket residues
Cofactor context
Docked ligand
Overall assessment
Weak No SASA yet
Weak or marginal quality
Binding strong Geometry high Native strong SASA missing
Strain ΔE
25.9 kcal/mol
Protein clashes
4
Internal clashes
1
Native overlap
contact recall 0.71, Jaccard 0.62, H-bond role recall 0.20
Burial
93%
Reason: no major geometry red flags detected
4 protein-contact clashes
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.717 kcal/mol/HA) ✓ Good fit quality (FQ -7.34) ✗ High strain energy (25.9 kcal/mol) ✗ Geometry warnings ✗ Minor protein-contact clashes (4) ✗ Many internal clashes (15) ℹ SASA not computed
Score
-26.521
kcal/mol
LE
-0.717
kcal/mol/HA
Fit Quality
-7.34
FQ (Leeson)
HAC
37
heavy atoms
MW
496
Da
LogP
3.01
cLogP
Strain ΔE
25.9 kcal/mol
SASA buried
computing…

Interaction summary

HB 1 HY 24 PI 2 CLASH 1
Final rank5.055Score-26.521
Inter norm-0.739Intra norm0.022
Top1000noExcludedno
Contacts18H-bonds1
Artifact reasongeometry warning; 15 clashes; 4 protein contact clashes; high strain Δ 34.1
Residues
ALA10 ARG29 ASN65 GLU31 ILE61 ILE8 LEU28 LEU68 NAP201 PHE32 PHE35 PRO27 PRO62 SER60 THR57 TYR122 VAL116 VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Receptor context

1 kept / 0 excluded
Receptor context filtering: interactions and SASA are computed against protein atoms plus allowed cofactors/ions. Native ligand-like HETATM partners are excluded from scoring.
Kept context 1 Excluded HETATM 0
Kept cofactors / ions
A:NAP201

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseHB0
IFP residues
ALA10 ASN65 ASP22 GLN36 GLU31 GLY117 GLY21 ILE61 ILE8 LEU23 LEU68 NAP201 PHE32 PHE35 PRO62 SER60 THR137 THR57 TYR122 VAL116 VAL9
Current overlap15Native recall0.71
Jaccard0.62RMSD-
HB strict1Strict recall0.20
HB same residue+role1HB role recall0.20
HB same residue1HB residue recall0.20

HB · H-bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

PI · π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

HY · Hydrophobic contacts

CLASH · Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBCTCT overlapCT recallHB role rec.RMSDExcluded
733 5.055222150773577 -0.739118 -26.5211 1 18 15 0.71 0.20 - no Current
745 5.375843873554705 -0.666012 -26.7132 1 18 15 0.71 0.00 - no Open
742 5.412367154325793 -0.684603 -18.0164 1 19 16 0.76 0.00 - no Open
753 5.672244631749802 -0.641938 -24.2542 0 18 15 0.71 0.00 - no Open
741 5.944365449117049 -0.647985 -19.1738 1 19 16 0.76 0.00 - no Open
746 6.116463099465139 -0.601075 -25.532 0 18 15 0.71 0.00 - no Open
743 6.135719338048507 -0.729853 -26.8143 0 19 16 0.76 0.00 - no Open
756 6.293183387382296 -0.721061 -29.3114 2 14 12 0.57 0.00 - no Open
749 6.583361142874363 -0.718459 -28.454 1 18 16 0.76 0.20 - no Open
751 6.657832340087772 -0.724408 -27.0298 0 20 17 0.81 0.00 - no Open
732 6.798701473728911 -0.727402 -22.3807 1 18 17 0.81 0.00 - no Open
731 6.873124190646189 -0.695817 -24.6461 1 17 14 0.67 0.20 - no Open
748 7.001076559763854 -0.658529 -26.6758 2 19 16 0.76 0.20 - no Open
327 7.0154060429700635 -0.412866 -11.6152 2 14 0 0.00 0.00 - no Open
539 7.583104340691228 -0.662156 -19.598 1 19 0 0.00 0.00 - no Open
740 7.7906750176752 -0.638331 -19.2618 1 20 17 0.81 0.20 - no Open
330 8.13830786553122 -0.284615 -9.20947 6 14 0 0.00 0.00 - no Open
542 8.28456516246071 -0.574589 -21.3313 1 13 0 0.00 0.00 - no Open
754 8.30935986735237 -0.641516 -28.7092 0 19 16 0.76 0.00 - no Open
750 8.48747499781867 -0.650881 -25.8966 1 19 15 0.71 0.00 - no Open
752 55.8025526412649 -0.749748 -24.7285 1 18 15 0.71 0.20 - no Open
735 7.75343195331093 -0.743617 -24.9413 1 20 17 0.81 0.00 - yes Open
734 8.064388656605804 -0.673188 -17.6561 1 18 14 0.67 0.00 - yes Open
738 9.113722165632222 -0.739701 -27.4729 2 18 18 0.86 0.20 - yes Open
541 9.147539801431252 -0.562609 -20.2124 1 18 0 0.00 0.00 - yes Open
755 9.509527302898046 -0.635604 -16.7201 1 18 15 0.71 0.00 - yes Open
736 9.826628313614366 -0.800981 -25.5375 1 19 17 0.81 0.20 - yes Open
329 9.892513973653447 -0.691497 -17.5451 7 16 0 0.00 0.00 - yes Open
739 10.876964291124517 -0.673595 -24.8894 1 15 12 0.57 0.00 - yes Open
324 12.094940289006843 -0.525789 -14.3441 6 17 0 0.00 0.00 - yes Open
325 12.567467433982564 -0.679503 -18.0868 5 16 0 0.00 0.00 - yes Open
326 13.212417045524774 -0.35492 7.41593 3 19 0 0.00 0.00 - yes Open
744 56.93641830148738 -0.639962 -25.4764 1 18 15 0.71 0.20 - yes Open
747 57.698358513556705 -0.666806 -21.7519 1 18 15 0.71 0.00 - yes Open
737 57.82255668118601 -0.778049 -24.9242 1 21 18 0.86 0.00 - yes Open
328 61.210501616092344 -0.432964 -12.0606 6 15 0 0.00 0.00 - yes Open
540 62.43049320007665 -0.600161 -18.1731 4 17 0 0.00 0.00 - yes Open
323 63.891854853100575 -0.243323 -0.609683 5 17 0 0.00 0.00 - yes Open

Molecular metrics

RDKit SASA burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -26.521kcal/mol
Ligand efficiency (LE) -0.7168kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.338
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 37HA

Physicochemical properties

Molecular weight 495.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.01
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 25.95kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 119.57kcal/mol
Minimised FF energy 93.62kcal/mol

SASA & burial

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate SASA burial metrics without blocking the page.