FAIRMol

NMT-TY0180

Pose ID 7165 Compound 870 Pose 578

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-2.213 kcal/mol/HA) ✓ Good fit quality (FQ -18.14) ✓ Good H-bonds (5 bonds) ✗ High strain energy (18.8 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-42.040
kcal/mol
LE
-2.213
kcal/mol/HA
Fit Quality
-18.14
FQ (Leeson)
HAC
19
heavy atoms
MW
276
Da
LogP
0.00
cLogP
Strain ΔE
18.8 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: mixed
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 18.8 kcal/mol

Interaction summary

Collapsible panels
H-bonds 5 Hydrophobic 16 π–π 2 Clashes 10 Severe clashes 0
Final rank4.5208806570532Score-42.0399
Inter norm-1.59846Intra norm-0.614167
Top1000noExcludedno
Contacts9H-bonds5
Artifact reasongeometry warning; 10 clashes; 10 protein contact clashes; very favorable intra outlier; high strain Δ 23.3
ResiduesA:ARG17;A:HIS241;A:LEU188;A:LEU226;A:LEU229;A:NDP302;A:PHE113;A:TYR194;D:ARG287

Protein summary

308 residues
Protein targetT04Atoms4210
Residues308Chains3
Residue summaryLEU:494; ALA:421; ARG:384; VAL:368; THR:295; TYR:231; SER:198; PRO:196; ILE:190; LYS:176; ASN:154; GLU:150; GLY:126; PHE:120; HIS:119; ASP:108

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name7PXXContacts19
PoseOpen native poseH-bonds8
IFP residuesA:ARG17; A:ASP181; A:GLY225; A:HIS241; A:LEU188; A:LEU226; A:LEU229; A:LYS198; A:MET233; A:NDP302; A:PHE113; A:PRO115; A:SER111; A:SER112; A:SER227; A:TYR191; A:TYR194; A:VAL230; D:ARG287
Current overlap9Native recall0.47
Jaccard0.47RMSD-
H-bond strict2Strict recall0.33
H-bond same residue+role2Role recall0.40
H-bond same residue3Residue recall0.60

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
582 3.499217272763817 -1.30109 -36.8386 6 11 11 0.58 0.60 - no Open
562 3.6187481355843296 -1.34079 -40.2599 6 10 10 0.53 0.60 - no Open
578 4.5208806570532 -1.59846 -42.0399 5 9 9 0.47 0.40 - no Current
570 5.209444608553848 -1.45307 -41.8283 6 10 10 0.53 0.40 - no Open
574 5.494287795351761 -1.19846 -34.3917 3 10 10 0.53 0.40 - no Open
576 7.10237483110608 -0.49952 -23.4625 6 13 12 0.63 0.40 - no Open
580 57.313683031445834 -1.03805 -35.4741 6 12 11 0.58 0.40 - no Open
564 5.683316417253755 -0.86167 -33.5312 2 11 11 0.58 0.00 - yes Open
569 6.688437061075931 -0.743094 -27.3628 1 11 11 0.58 0.00 - yes Open
584 7.470859734600507 -1.01745 -32.0466 7 12 11 0.58 0.60 - yes Open
563 7.597906003760038 -0.936069 -26.9598 9 9 9 0.47 0.60 - yes Open
583 7.71554455855693 -1.04816 -29.2323 9 9 9 0.47 0.60 - yes Open
568 7.8494213242796524 -0.88423 -32.0146 2 11 11 0.58 0.00 - yes Open
577 55.44856952842226 -0.737756 -26.3696 1 11 11 0.58 0.00 - yes Open
581 55.82706248093621 -0.957868 -10.4022 8 11 11 0.58 0.40 - yes Open
565 57.12469603240336 -1.01851 -28.9888 7 10 10 0.53 0.40 - yes Open
579 57.35827406946044 -1.20655 -31.9233 8 9 9 0.47 0.40 - yes Open
567 58.30396694034117 -0.848766 -27.2641 8 9 9 0.47 0.40 - yes Open
572 58.527859333387774 -1.05053 -28.9048 6 10 10 0.53 0.60 - yes Open
575 58.81464145758146 -0.837151 -27.0263 6 13 13 0.68 0.40 - yes Open
571 58.81822193260073 -1.13201 -32.3157 8 9 9 0.47 0.40 - yes Open
566 59.028973574358915 -0.671315 -27.8576 0 11 11 0.58 0.00 - yes Open
585 60.22855226760838 -0.895668 -29.5255 7 10 10 0.53 0.40 - yes Open
573 60.428095187948756 -0.886832 -24.3607 9 9 9 0.47 0.40 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -42.040kcal/mol
Ligand efficiency (LE) -2.2126kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -18.136
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 19HA

Physicochemical properties

Molecular weight 276.3Da
Lipinski: ≤ 500 Da
LogP (cLogP) 0.00
Lipinski: ≤ 5
Rotatable bonds 1

Conformational strain (MMFF94s)

Strain energy (ΔE) 18.80kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 56.25kcal/mol
Minimised FF energy 37.45kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.