FAIRMol

KB_Leish_46

Pose ID 702 Compound 143 Pose 702

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.592 kcal/mol/HA) ✓ Good fit quality (FQ -5.82) ✓ Good H-bonds (3 bonds) ✗ Very high strain energy (27.7 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-18.934
kcal/mol
LE
-0.592
kcal/mol/HA
Fit Quality
-5.82
FQ (Leeson)
HAC
32
heavy atoms
MW
478
Da
LogP
3.61
cLogP
Strain ΔE
27.7 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 27.7 kcal/mol

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 24 π–π 1 Clashes 9 Severe clashes 0
Final rank6.237814060192159Score-18.9343
Inter norm-0.818133Intra norm0.226435
Top1000noExcludedno
Contacts18H-bonds3
Artifact reasongeometry warning; 15 clashes; 9 protein contact clashes; high strain Δ 31.0
ResiduesA:ALA10;A:ASN65;A:ASP22;A:GLN36;A:GLU31;A:GLY21;A:ILE61;A:ILE8;A:LEU23;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO62;A:SER60;A:THR57;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap18Native recall0.86
Jaccard0.86RMSD-
H-bond strict1Strict recall0.20
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
686 4.213267745548484 -0.802746 -25.7539 0 19 16 0.76 0.00 - no Open
700 4.220010643766157 -0.832652 -28.5179 2 20 19 0.90 0.20 - no Open
682 4.570105105839405 -0.625261 -21.3428 2 15 13 0.62 0.20 - no Open
684 5.0874575879674655 -0.818542 -25.5255 2 21 19 0.90 0.20 - no Open
702 6.237814060192159 -0.818133 -18.9343 3 18 18 0.86 0.20 - no Current
704 6.492055677533312 -0.814606 -26.1757 4 21 19 0.90 0.00 - no Open
683 54.257864021424815 -0.65648 -23.8839 1 17 16 0.76 0.20 - yes Open
698 54.845749901123966 -0.745182 -23.6958 2 20 19 0.90 0.20 - yes Open
688 55.49278811701789 -0.800433 -24.8696 1 19 17 0.81 0.20 - yes Open
693 56.41654722764329 -0.633508 -14.5988 2 13 12 0.57 0.00 - yes Open
696 56.880054504002274 -0.705585 -19.6321 1 16 15 0.71 0.00 - yes Open
697 57.151250079463736 -0.80801 -22.4749 2 18 16 0.76 0.00 - yes Open
694 57.15309101774906 -0.839171 -29.6744 5 19 17 0.81 0.20 - yes Open
690 57.242661857823634 -0.666712 -14.1732 2 19 15 0.71 0.20 - yes Open
685 57.746874096747156 -0.746492 -24.1771 2 19 17 0.81 0.00 - yes Open
692 58.10140529217655 -0.756074 -23.3523 2 21 19 0.90 0.20 - yes Open
691 58.14232666846858 -0.69608 -18.0573 2 16 13 0.62 0.00 - yes Open
699 58.83392169415286 -0.752237 -23.925 3 16 15 0.71 0.00 - yes Open
681 59.12171868342816 -0.77085 -25.1165 2 14 11 0.52 0.00 - yes Open
687 59.467111024549816 -0.686365 -18.4284 2 19 16 0.76 0.00 - yes Open
701 60.57259410637262 -0.713888 -21.5699 2 17 15 0.71 0.00 - yes Open
689 61.35090917829254 -0.731009 -22.7288 2 21 18 0.86 0.00 - yes Open
703 61.89591576324208 -0.675811 -22.8023 2 19 17 0.81 0.00 - yes Open
695 62.47334985863181 -0.705648 -21.8198 2 20 18 0.86 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -18.934kcal/mol
Ligand efficiency (LE) -0.5917kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -5.819
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 32HA

Physicochemical properties

Molecular weight 478.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.61
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 27.69kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 60.08kcal/mol
Minimised FF energy 32.40kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.