FAIRMol

ulfkktlib_1309

Pose ID 6902 Compound 913 Pose 315

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-1.051 kcal/mol/HA) ✓ Good fit quality (FQ -9.28) ✓ Good H-bonds (4 bonds) ✗ Very high strain energy (29.1 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-24.182
kcal/mol
LE
-1.051
kcal/mol/HA
Fit Quality
-9.28
FQ (Leeson)
HAC
23
heavy atoms
MW
340
Da
LogP
1.99
cLogP
Strain ΔE
29.1 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 29.1 kcal/mol

Interaction summary

Collapsible panels
H-bonds 4 Hydrophobic 20 π–π 2 Clashes 11 Severe clashes 1
Final rank6.247149360892461Score-24.1822
Inter norm-1.22035Intra norm0.168955
Top1000noExcludedyes
Contacts13H-bonds4
Artifact reasonexcluded; geometry warning; 7 clashes; 1 protein clash; high strain Δ 29.6
ResiduesA:ARG17;A:GLY225;A:HIS241;A:LEU188;A:LEU226;A:LEU229;A:MET233;A:NDP302;A:PHE113;A:SER111;A:TYR191;A:TYR194;D:ARG287

Protein summary

308 residues
Protein targetT04Atoms4210
Residues308Chains3
Residue summaryLEU:494; ALA:421; ARG:384; VAL:368; THR:295; TYR:231; SER:198; PRO:196; ILE:190; LYS:176; ASN:154; GLU:150; GLY:126; PHE:120; HIS:119; ASP:108

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name7PXXContacts19
PoseOpen native poseH-bonds8
IFP residuesA:ARG17; A:ASP181; A:GLY225; A:HIS241; A:LEU188; A:LEU226; A:LEU229; A:LYS198; A:MET233; A:NDP302; A:PHE113; A:PRO115; A:SER111; A:SER112; A:SER227; A:TYR191; A:TYR194; A:VAL230; D:ARG287
Current overlap13Native recall0.68
Jaccard0.68RMSD-
H-bond strict1Strict recall0.17
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
316 3.993609952448017 -1.0862 -21.85 4 9 9 0.47 0.20 - no Open
314 4.097751272796711 -1.07406 -24.398 5 10 10 0.53 0.20 - no Open
313 5.267864876150979 -1.05033 -13.5139 3 13 13 0.68 0.20 - yes Open
315 6.247149360892461 -1.22035 -24.1822 4 13 13 0.68 0.20 - yes Current

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -24.182kcal/mol
Ligand efficiency (LE) -1.0514kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -9.279
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 23HA

Physicochemical properties

Molecular weight 339.8Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.99
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 29.13kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 37.57kcal/mol
Minimised FF energy 8.45kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.