FAIRMol

Z45925616

Pose ID 6189 Compound 544 Pose 2871

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.882 kcal/mol/HA) ✓ Good fit quality (FQ -8.33) ✗ Very high strain energy (23.4 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-24.698
kcal/mol
LE
-0.882
kcal/mol/HA
Fit Quality
-8.33
FQ (Leeson)
HAC
28
heavy atoms
MW
407
Da
LogP
5.83
cLogP
Strain ΔE
23.4 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 23.4 kcal/mol

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 24 π–π 4 Clashes 6 Severe clashes 2
Final rank7.10882567693303Score-24.6981
Inter norm-0.986494Intra norm0.10442
Top1000noExcludedyes
Contacts17H-bonds2
Artifact reasonexcluded; geometry warning; 13 clashes; 2 protein clashes; high strain Δ 28.1
ResiduesA:ALA32;A:ARG48;A:ARG97;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:LYS95;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:THR180;A:TRP47;A:VAL30;A:VAL31;A:VAL49

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap13Native recall0.65
Jaccard0.54RMSD-
H-bond strict1Strict recall0.14
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2043 2.9963607481740455 -0.870322 -27.6293 3 18 1 0.05 0.00 - no Open
1909 3.689900294712992 -0.801575 -22.6751 4 12 0 0.00 0.00 - no Open
2326 3.705716829060318 -0.577223 -16.6977 2 9 0 0.00 0.00 - no Open
2870 4.050305824450855 -0.790025 -23.2398 3 11 9 0.45 0.00 - no Open
2044 5.069101694248104 -0.797811 -23.0137 2 14 1 0.05 0.00 - no Open
3464 5.702951618806277 -0.760193 -17.1572 2 13 0 0.00 0.00 - no Open
3625 6.284865441525752 -0.735557 -21.605 1 13 0 0.00 0.00 - no Open
3463 6.415741126707506 -0.828835 -18.3728 2 16 0 0.00 0.00 - no Open
3627 6.663919820193825 -0.749836 -23.5599 2 11 1 0.05 0.00 - no Open
2327 5.201536113397625 -0.669419 -17.579 3 12 0 0.00 0.00 - yes Open
2045 5.778366047235093 -0.693995 -21.3166 1 16 1 0.05 0.00 - yes Open
2046 6.1878097351617845 -0.74483 -22.2983 2 15 1 0.05 0.00 - yes Open
1907 6.216464626402162 -0.914844 -25.1026 4 13 0 0.00 0.00 - yes Open
3465 6.270855112040639 -0.784948 -21.9872 1 15 0 0.00 0.00 - yes Open
3628 6.402791360590602 -0.694176 -19.7207 4 14 1 0.05 0.00 - yes Open
3626 6.622495608429628 -0.807393 -24.035 2 16 0 0.00 0.00 - yes Open
2328 6.820727394998152 -0.564702 -17.1982 2 10 0 0.00 0.00 - yes Open
2871 7.10882567693303 -0.986494 -24.6981 2 17 13 0.65 0.20 - yes Current
3462 7.162171496558556 -0.789896 -19.4096 3 17 0 0.00 0.00 - yes Open
2868 7.791682645393914 -0.851972 -20.1413 4 18 14 0.70 0.40 - yes Open
2869 8.288375686376511 -1.06292 -27.7872 2 16 13 0.65 0.20 - yes Open
1908 8.699957135349466 -0.783758 -15.2456 2 17 0 0.00 0.00 - yes Open
1910 9.791668457905187 -0.727799 -12.3201 3 17 0 0.00 0.00 - yes Open
2329 11.561716334351372 -0.596354 -14.53 3 8 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -24.698kcal/mol
Ligand efficiency (LE) -0.8821kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -8.327
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 28HA

Physicochemical properties

Molecular weight 406.9Da
Lipinski: ≤ 500 Da
LogP (cLogP) 5.83
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 23.38kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 78.78kcal/mol
Minimised FF energy 55.40kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.