FAIRMol

Z31287542

Pose ID 6172 Compound 745 Pose 2854

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.836 kcal/mol/HA) ✓ Good fit quality (FQ -8.37) ✓ Good H-bonds (3 bonds) ✗ Very high strain energy (29.5 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-28.425
kcal/mol
LE
-0.836
kcal/mol/HA
Fit Quality
-8.37
FQ (Leeson)
HAC
34
heavy atoms
MW
476
Da
LogP
3.33
cLogP
Strain ΔE
29.5 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 29.5 kcal/mol

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 24 π–π 3 Clashes 10 Severe clashes 4
Final rank13.695905445005074Score-28.4251
Inter norm-0.777668Intra norm-0.0583628
Top1000noExcludedyes
Contacts13H-bonds3
Artifact reasonexcluded; geometry warning; 24 clashes; 4 protein clashes; high strain Δ 41.7
ResiduesA:ALA32;A:ARG97;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:LYS95;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:THR54;A:VAL31

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap12Native recall0.60
Jaccard0.57RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1514 7.533781901841193 -0.634882 -21.4916 2 12 0 0.00 0.00 - no Open
1519 7.946048041711834 -0.337285 -12.4181 0 12 0 0.00 0.00 - no Open
1516 8.037752732679447 -0.832101 -28.9631 1 13 0 0.00 0.00 - no Open
2852 8.48620637071585 -0.831972 -28.6804 2 18 14 0.70 0.20 - no Open
1583 9.232988641186012 -0.94457 -33.9929 6 19 0 0.00 0.00 - no Open
2859 8.441706828631817 -0.587213 -21.1824 0 14 11 0.55 0.00 - yes Open
1518 8.546547835918052 -0.85907 -28.691 2 12 0 0.00 0.00 - yes Open
1520 8.565928211114365 -0.5023 -13.6734 2 12 0 0.00 0.00 - yes Open
2858 8.61612676343768 -0.675324 -23.4232 2 13 10 0.50 0.20 - yes Open
1515 8.800782866793854 -0.706498 -24.139 3 10 0 0.00 0.00 - yes Open
1584 9.137800022550554 -0.902122 -29.855 4 20 0 0.00 0.00 - yes Open
2856 9.22048295162044 -0.754895 -24.7354 0 17 13 0.65 0.00 - yes Open
1586 9.221161529299227 -0.703799 -25.1048 9 5 0 0.00 0.00 - yes Open
2853 10.330473319524868 -0.645165 -22.0761 3 19 15 0.75 0.00 - yes Open
2854 13.695905445005074 -0.777668 -28.4251 3 13 12 0.60 0.00 - yes Current
1585 58.98715940547089 -0.876248 -31.2541 6 22 0 0.00 0.00 - yes Open
1517 58.99014428676841 -0.436484 -11.9302 1 15 0 0.00 0.00 - yes Open
2857 59.549788082864985 -0.834785 -25.7247 4 14 13 0.65 0.20 - yes Open
2855 62.18538355187409 -0.659105 -21.5791 3 13 9 0.45 0.20 - yes Open
1521 62.87410528533428 -0.498737 -17.4697 3 12 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -28.425kcal/mol
Ligand efficiency (LE) -0.8360kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -8.365
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 34HA

Physicochemical properties

Molecular weight 475.9Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.33
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 29.48kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 124.93kcal/mol
Minimised FF energy 95.45kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.