FAIRMol

Z49542045

Pose ID 6082 Compound 735 Pose 2764

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.873 kcal/mol/HA) ✓ Good fit quality (FQ -8.51) ✓ Good H-bonds (4 bonds) ✗ Very high strain energy (58.5 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-27.064
kcal/mol
LE
-0.873
kcal/mol/HA
Fit Quality
-8.51
FQ (Leeson)
HAC
31
heavy atoms
MW
442
Da
LogP
3.53
cLogP
Strain ΔE
58.5 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 58.5 kcal/mol

Interaction summary

Collapsible panels
H-bonds 4 Hydrophobic 24 π–π 3 Clashes 9 Severe clashes 0
Final rank7.7517023364703235Score-27.0636
Inter norm-0.851646Intra norm-0.0213748
Top1000noExcludedno
Contacts19H-bonds4
Artifact reasongeometry warning; 14 clashes; 9 protein contact clashes; high strain Δ 59.6
ResiduesA:ALA32;A:ARG97;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:LYS95;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:PRO93;A:THR180;A:THR83;A:TYR162;A:VAL156;A:VAL30;A:VAL31;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap17Native recall0.85
Jaccard0.77RMSD-
H-bond strict1Strict recall0.14
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1356 7.30919015569561 -0.747819 -22.4692 4 12 0 0.00 0.00 - no Open
2766 7.626560514791622 -0.76421 -21.2192 4 14 14 0.70 0.20 - no Open
2764 7.7517023364703235 -0.851646 -27.0636 4 19 17 0.85 0.20 - no Current
1354 8.091391784310396 -0.76201 -22.4584 3 13 0 0.00 0.00 - no Open
1357 8.286357705039862 -0.71293 -20.1897 1 15 0 0.00 0.00 - no Open
1358 8.509331768833594 -0.765906 -22.5045 3 11 0 0.00 0.00 - no Open
1673 8.575978773607371 -0.953186 -27.6149 8 15 0 0.00 0.00 - no Open
1669 8.816759867335094 -1.03081 -29.7112 9 15 0 0.00 0.00 - no Open
1672 9.362017157837828 -0.97062 -23.9871 8 18 0 0.00 0.00 - no Open
1353 9.570110861770155 -0.762672 -21.9133 2 15 0 0.00 0.00 - yes Open
1670 9.58932627039659 -0.902423 -27.2893 8 17 0 0.00 0.00 - yes Open
1668 9.675499203019521 -0.847302 -21.3097 7 17 0 0.00 0.00 - yes Open
1355 9.982986083410468 -0.647251 -16.8308 3 12 0 0.00 0.00 - yes Open
2768 11.772406665392056 -0.812859 -20.601 5 14 10 0.50 0.20 - yes Open
2765 13.036634138808747 -0.69553 -21.8898 3 14 9 0.45 0.20 - yes Open
2767 14.005140975277962 -0.649309 -18.2469 3 14 13 0.65 0.20 - yes Open
2763 14.712984028568691 -0.74996 -16.6372 4 13 9 0.45 0.20 - yes Open
1671 16.875902029159732 -0.928572 -27.141 7 17 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -27.064kcal/mol
Ligand efficiency (LE) -0.8730kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -8.505
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 31HA

Physicochemical properties

Molecular weight 442.5Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.53
Lipinski: ≤ 5
Rotatable bonds 8

Conformational strain (MMFF94s)

Strain energy (ΔE) 58.45kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 101.55kcal/mol
Minimised FF energy 43.09kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.