FAIRMol

Z47741866

Pose ID 6079 Compound 513 Pose 2761

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing
T03
Bifunctional dihydrofolate reductase-thymidylate synthase (DHFR-TS) 'ambiguous: archive label suggests Leishmania major, structure title points to Trypanosoma cruzi template'
Ligand Z47741866
PDB3CL9

3D complex viewer

Strict H-bonds Permissive H-bonds
Viewer legend
Protein receptor
Pocket residues
Cofactor context
Docked ligand
Overall assessment
Reject No SASA yet
Promising but geometrically suspicious
Binding strong Geometry low Native strong SASA missing
Strain ΔE
24.1 kcal/mol
Protein clashes
5
Internal clashes
10
Native overlap
contact recall 0.65, Jaccard 0.57, H-bond role recall 0.80
Burial
94%
Reason: 10 internal clashes
5 protein-contact clashes 10 intramolecular clashes
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.991 kcal/mol/HA) ✓ Good fit quality (FQ -9.13) ✓ Strong H-bond network (8 bonds) ✗ High strain energy (24.1 kcal/mol) ✗ Geometry warnings ✗ Protein-contact clashes (5) ✗ Many internal clashes (10) ℹ SASA not computed
Score
-25.774
kcal/mol
LE
-0.991
kcal/mol/HA
Fit Quality
-9.13
FQ (Leeson)
HAC
26
heavy atoms
MW
369
Da
LogP
2.83
cLogP
Strain ΔE
24.1 kcal/mol
SASA buried
computing…

Interaction summary

HB 8 HY 24 PI 1 CLASH 0
Final rank3.680Score-25.774
Inter norm-1.114Intra norm0.123
Top1000noExcludedno
Contacts16H-bonds8
Artifact reasongeometry warning; 10 clashes; 5 protein contact clashes; high strain Δ 27.1
Residues
ALA32 ARG48 ARG97 ASP52 ILE45 LEU94 LYS57 MET53 NDP301 PHE56 PHE91 TRP47 TYR162 VAL30 VAL31 VAL49

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Receptor context

1 kept / 0 excluded
Receptor context filtering: interactions and SASA are computed against protein atoms plus allowed cofactors/ions. Native ligand-like HETATM partners are excluded from scoring.
Kept context 1 Excluded HETATM 0
Kept cofactors / ions
A:NDP301

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseHB0
IFP residues
ALA32 ARG97 ASP52 ILE45 LEU94 LYS57 MET53 NDP301 PHE56 PHE91 PRO88 SER86 THR180 THR54 THR83 TYR162 VAL156 VAL30 VAL31 VAL87
Current overlap13Native recall0.65
Jaccard0.57RMSD-
HB strict4Strict recall0.57
HB same residue+role4HB role recall0.80
HB same residue4HB residue recall0.80

HB · H-bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

PI · π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

HY · Hydrophobic contacts

CLASH · Clashes

No clash · clashes detected for this pose.

All stored poses for this docking hit

PoseFinal rankInter normScoreHBCTCT overlapCT recallHB role rec.RMSDExcluded
2761 3.679571422655938 -1.1141 -25.774 8 16 13 0.65 0.80 - no Current
2015 3.9637882795787753 -0.708788 -16.62 7 10 0 0.00 0.00 - no Open
1783 4.50899255342546 -0.950014 -21.6522 6 14 0 0.00 0.00 - no Open
3392 5.024280167565795 -0.760226 -18.4075 2 14 0 0.00 0.00 - no Open
2016 5.249917048313938 -0.868198 -19.1442 8 11 0 0.00 0.00 - no Open
3393 5.836985889792018 -0.931065 -21.7495 6 17 0 0.00 0.00 - no Open
1784 4.8360261066062575 -1.03976 -24.8291 5 19 0 0.00 0.00 - yes Open
2762 9.507763869675289 -0.946253 -22.0577 7 15 11 0.55 0.40 - yes Open

Molecular metrics

RDKit SASA burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -25.774kcal/mol
Ligand efficiency (LE) -0.9913kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -9.133
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 26HA

Physicochemical properties

Molecular weight 369.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.83
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 24.05kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 34.98kcal/mol
Minimised FF energy 10.92kcal/mol

SASA & burial

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate SASA burial metrics without blocking the page.