FAIRMol

Z56935963

Pose ID 6029 Compound 547 Pose 2711

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-1.078 kcal/mol/HA) ✓ Good fit quality (FQ -9.93) ✓ Good H-bonds (5 bonds) ✗ Very high strain energy (34.0 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-28.019
kcal/mol
LE
-1.078
kcal/mol/HA
Fit Quality
-9.93
FQ (Leeson)
HAC
26
heavy atoms
MW
391
Da
LogP
2.82
cLogP
Strain ΔE
34.0 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 34.0 kcal/mol

Interaction summary

Collapsible panels
H-bonds 5 Hydrophobic 17 π–π 2 Clashes 9 Severe clashes 0
Final rank5.671810626257038Score-28.0194
Inter norm-0.730073Intra norm-0.347597
Top1000noExcludedno
Contacts16H-bonds5
Artifact reasongeometry warning; 7 clashes; 9 protein contact clashes; very favorable intra outlier; high strain Δ 44.1
ResiduesA:ARG48;A:ARG97;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:PRO88;A:THR83;A:TRP47;A:VAL156;A:VAL49;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap13Native recall0.65
Jaccard0.57RMSD-
H-bond strict1Strict recall0.14
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
3351 3.700166410105763 -0.694355 -24.1012 7 12 0 0.00 0.00 - no Open
3356 4.060259190723226 -0.57646 -16.2213 5 15 0 0.00 0.00 - no Open
2708 4.066908340758205 -0.882299 -23.5614 7 19 14 0.70 0.20 - no Open
2713 4.397339357329831 -0.882041 -26.1356 7 9 7 0.35 0.20 - no Open
3357 4.52185972612399 -0.614849 -12.8325 3 12 0 0.00 0.00 - no Open
2721 4.600408778455224 -0.734888 -14.8762 8 18 13 0.65 0.00 - no Open
2709 4.8485224772625015 -1.05932 -24.7891 6 17 14 0.70 0.20 - no Open
2722 4.94558020240054 -0.817679 -21.4264 4 17 13 0.65 0.00 - no Open
2716 4.9667622754639424 -0.825218 -24.6944 6 17 14 0.70 0.20 - no Open
3347 5.520272521802061 -0.783828 -21.1306 8 11 0 0.00 0.00 - no Open
2711 5.671810626257038 -0.730073 -28.0194 5 16 13 0.65 0.20 - no Current
3343 4.907718538764667 -0.926049 -23.919 8 12 0 0.00 0.00 - yes Open
3355 5.327273340927074 -0.804704 -22.4335 7 14 0 0.00 0.00 - yes Open
2717 5.51011414711577 -0.80878 -22.5146 2 19 15 0.75 0.00 - yes Open
3348 5.535934980262025 -0.922918 -24.4857 6 15 0 0.00 0.00 - yes Open
3352 5.967136058308274 -0.615596 -19.4533 5 11 0 0.00 0.00 - yes Open
2714 6.03655169233735 -0.825675 -22.2478 6 14 11 0.55 0.20 - yes Open
3353 6.388856661844819 -0.711742 -18.4431 6 12 0 0.00 0.00 - yes Open
2712 6.455154962785032 -0.883812 -24.8654 4 17 14 0.70 0.00 - yes Open
3349 6.512434389319291 -0.694102 -20.8902 7 14 0 0.00 0.00 - yes Open
3346 7.02004168331491 -0.681302 -27.0085 3 14 0 0.00 0.00 - yes Open
2719 7.518280240178267 -0.766525 -20.3131 2 17 15 0.75 0.00 - yes Open
2723 7.537187184503247 -0.751544 -18.5869 6 14 11 0.55 0.20 - yes Open
3345 8.74043112610656 -0.721575 -19.8508 4 14 0 0.00 0.00 - yes Open
2715 55.78029250972965 -0.834686 -21.8621 4 14 10 0.50 0.00 - yes Open
3350 55.941164464406576 -0.62208 -19.4593 3 10 0 0.00 0.00 - yes Open
3358 56.52519508621056 -0.700347 -20.783 6 13 0 0.00 0.00 - yes Open
2720 57.276901634848244 -0.858543 -23.2142 6 17 14 0.70 0.20 - yes Open
2710 57.34572465987451 -1.00114 -24.3262 6 16 13 0.65 0.20 - yes Open
3344 57.94765240802333 -0.74487 -23.0944 8 10 0 0.00 0.00 - yes Open
3354 58.007845546614455 -0.811484 -21.7359 5 14 0 0.00 0.00 - yes Open
2718 58.43349222570747 -0.970525 -25.3633 6 14 10 0.50 0.20 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -28.019kcal/mol
Ligand efficiency (LE) -1.0777kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -9.929
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 26HA

Physicochemical properties

Molecular weight 391.5Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.82
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 34.03kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 113.69kcal/mol
Minimised FF energy 79.66kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.