FAIRMol

Z56773052

Pose ID 5841 Compound 507 Pose 2523

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.575 kcal/mol/HA) ✓ Good fit quality (FQ -5.42) ✓ Good H-bonds (3 bonds) ✗ Very high strain energy (23.0 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-16.087
kcal/mol
LE
-0.575
kcal/mol/HA
Fit Quality
-5.42
FQ (Leeson)
HAC
28
heavy atoms
MW
406
Da
LogP
5.56
cLogP
Strain ΔE
23.0 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 23.0 kcal/mol

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 23 π–π 3 Clashes 14 Severe clashes 2
Final rank8.472204082026884Score-16.0871
Inter norm-0.938303Intra norm0.363763
Top1000noExcludedyes
Contacts14H-bonds3
Artifact reasonexcluded; geometry warning; 8 clashes; 2 protein clashes; high strain Δ 23.0
ResiduesA:ALA32;A:ARG97;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:LYS95;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:TYR162;A:VAL30;A:VAL31

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap13Native recall0.65
Jaccard0.62RMSD-
H-bond strict2Strict recall0.29
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2522 3.603100088384475 -0.753208 -20.2271 1 15 13 0.65 0.00 - no Open
1046 4.115524958213157 -0.877037 -21.4858 1 11 0 0.00 0.00 - no Open
1045 4.334165538881587 -0.924931 -23.7852 1 11 0 0.00 0.00 - no Open
1048 4.664008092419392 -0.82573 -20.6883 1 12 0 0.00 0.00 - no Open
2524 4.874806654884296 -0.773568 -21.3083 1 15 13 0.65 0.00 - no Open
1047 5.052657343141703 -0.898838 -21.5124 1 11 0 0.00 0.00 - no Open
1567 5.509606217872089 -0.912214 -16.18 4 20 1 0.05 0.00 - no Open
1566 5.372919973915165 -0.7248 -19.5067 2 12 1 0.05 0.00 - yes Open
1568 5.79009765527818 -0.701841 -20.5574 3 12 1 0.05 0.00 - yes Open
1569 6.581816602297611 -0.837093 -14.3369 1 20 1 0.05 0.00 - yes Open
2521 7.828736633834243 -0.957989 -17.416 4 14 13 0.65 0.20 - yes Open
2523 8.472204082026884 -0.938303 -16.0871 3 14 13 0.65 0.20 - yes Current

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -16.087kcal/mol
Ligand efficiency (LE) -0.5745kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -5.424
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 28HA

Physicochemical properties

Molecular weight 405.9Da
Lipinski: ≤ 500 Da
LogP (cLogP) 5.56
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 23.02kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 77.19kcal/mol
Minimised FF energy 54.17kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.