FAIRMol

KB_HAT_92

Pose ID 576 Compound 229 Pose 576

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.727 kcal/mol/HA) ✓ Good fit quality (FQ -7.21) ✗ Very high strain energy (22.6 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-23.991
kcal/mol
LE
-0.727
kcal/mol/HA
Fit Quality
-7.21
FQ (Leeson)
HAC
33
heavy atoms
MW
468
Da
LogP
4.19
cLogP
Strain ΔE
22.6 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 22.6 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 1 Clashes 6 Severe clashes 0
Final rank4.899166227216967Score-23.9915
Inter norm-0.814986Intra norm0.0879715
Top1000noExcludedno
Contacts16H-bonds1
Artifact reasongeometry warning; 13 clashes; 6 protein contact clashes; high strain Δ 31.3
ResiduesA:ALA10;A:ASP22;A:GLU31;A:GLY21;A:ILE8;A:LEU23;A:NAP201;A:PHE32;A:PHE35;A:PRO26;A:PRO27;A:SER60;A:TRP25;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap13Native recall0.62
Jaccard0.54RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
576 4.899166227216967 -0.814986 -23.9915 1 16 13 0.62 0.00 - no Current
585 5.051291435012429 -0.606897 -20.4888 1 15 14 0.67 0.00 - no Open
582 5.0678324087449 -0.789528 -26.2562 1 18 15 0.71 0.00 - no Open
583 5.211303678384479 -0.786735 -26.4341 1 18 15 0.71 0.00 - no Open
571 5.675978054170416 -0.749573 -22.4422 1 18 15 0.71 0.00 - no Open
575 6.509177088044854 -0.749189 -22.444 1 20 16 0.76 0.00 - no Open
581 55.5472851665849 -0.722467 -23.9796 2 18 14 0.67 0.00 - no Open
573 56.24336170495873 -0.748887 -24.6343 2 17 14 0.67 0.00 - no Open
578 54.9835115075708 -0.773782 -23.0825 2 19 16 0.76 0.00 - yes Open
584 55.293739389465806 -0.689029 -23.9432 2 14 13 0.62 0.00 - yes Open
574 55.87361695408371 -0.778508 -25.4926 2 18 15 0.71 0.00 - yes Open
572 56.71683154578473 -0.665379 -23.9974 2 18 14 0.67 0.20 - yes Open
577 57.73266711400078 -0.698289 -24.0488 2 16 12 0.57 0.20 - yes Open
586 58.27048055040028 -0.758645 -23.331 2 16 15 0.71 0.00 - yes Open
579 58.40335435533965 -0.718755 -23.7303 2 16 14 0.67 0.00 - yes Open
580 61.606000420482786 -0.742052 -23.5076 5 20 18 0.86 0.40 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -23.991kcal/mol
Ligand efficiency (LE) -0.7270kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.213
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 33HA

Physicochemical properties

Molecular weight 467.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 4.19
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 22.58kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 31.43kcal/mol
Minimised FF energy 8.85kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.