FAIRMol

MK178

Pose ID 5492 Compound 138 Pose 2174

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-1.040 kcal/mol/HA) ✓ Good fit quality (FQ -9.70) ✓ Strong H-bond network (7 bonds) ✗ Very high strain energy (25.3 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-28.074
kcal/mol
LE
-1.040
kcal/mol/HA
Fit Quality
-9.70
FQ (Leeson)
HAC
27
heavy atoms
MW
384
Da
LogP
-0.23
cLogP
Strain ΔE
25.3 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 25.3 kcal/mol

Interaction summary

Collapsible panels
H-bonds 7 Hydrophobic 20 π–π 2 Clashes 9 Severe clashes 2
Final rank7.548052921400164Score-28.0737
Inter norm-1.00177Intra norm-0.0379968
Top1000noExcludedyes
Contacts17H-bonds7
Artifact reasonexcluded; geometry warning; 10 clashes; 2 protein clashes; high strain Δ 28.9
ResiduesA:ALA32;A:ARG97;A:GLY157;A:ILE45;A:LEU94;A:LYS57;A:LYS95;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:PRO93;A:TYR162;A:VAL156;A:VAL30;A:VAL31;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap14Native recall0.70
Jaccard0.61RMSD-
H-bond strict3Strict recall0.43
H-bond same residue+role3Role recall0.60
H-bond same residue3Residue recall0.60

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2173 3.8345008776306306 -0.937733 -26.8154 7 18 16 0.80 0.60 - no Open
2084 4.198712269445888 -1.00925 -27.9623 4 17 0 0.00 0.00 - no Open
1064 4.226444352922489 -0.949988 -21.439 9 18 1 0.05 0.00 - no Open
1321 4.463774663390536 -0.745014 -17.1304 6 12 0 0.00 0.00 - no Open
1581 4.764200594088818 -0.761878 -19.574 5 14 0 0.00 0.00 - no Open
2172 5.292143248216333 -1.03355 -25.1287 8 15 13 0.65 0.80 - no Open
752 7.178404730818723 -1.12639 -29.0563 5 19 0 0.00 0.00 - no Open
1322 5.9536044379003865 -0.739406 -18.7461 5 11 0 0.00 0.00 - yes Open
2171 7.316161169363361 -0.998196 -27.7984 7 17 15 0.75 0.80 - yes Open
1065 7.516959271657992 -1.0482 -25.1368 8 17 1 0.05 0.00 - yes Open
2174 7.548052921400164 -1.00177 -28.0737 7 17 14 0.70 0.60 - yes Current
1320 9.439912653943008 -0.883222 -24.6464 5 14 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -28.074kcal/mol
Ligand efficiency (LE) -1.0398kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -9.701
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 27HA

Physicochemical properties

Molecular weight 384.5Da
Lipinski: ≤ 500 Da
LogP (cLogP) -0.23
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 25.33kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 47.28kcal/mol
Minimised FF energy 21.95kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.