FAIRMol

TC392

Pose ID 5382 Compound 107 Pose 2064

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.902 kcal/mol/HA) ✓ Good fit quality (FQ -8.70) ✓ Good H-bonds (5 bonds) ✗ High strain energy (11.2 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-27.051
kcal/mol
LE
-0.902
kcal/mol/HA
Fit Quality
-8.70
FQ (Leeson)
HAC
30
heavy atoms
MW
429
Da
LogP
4.30
cLogP
Strain ΔE
11.2 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: mixed
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 11.2 kcal/mol

Interaction summary

Collapsible panels
H-bonds 5 Hydrophobic 24 π–π 2 Clashes 8 Severe clashes 2
Final rank6.977560368249202Score-27.0509
Inter norm-0.921564Intra norm0.0198669
Top1000noExcludedyes
Contacts15H-bonds5
Artifact reasonexcluded; geometry warning; 12 clashes; 2 protein clashes; moderate strain Δ 14.7
ResiduesA:ALA32;A:ARG48;A:ARG97;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:LYS95;A:MET53;A:PHE56;A:PHE91;A:PRO93;A:TRP47;A:VAL49;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap10Native recall0.50
Jaccard0.40RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2065 2.94602425672637 -0.992564 -28.8915 4 18 16 0.80 0.20 - no Open
1191 3.768089679049951 -0.719092 -19.5389 5 14 0 0.00 0.00 - no Open
1962 3.9333827126534873 -0.900549 -22.9333 4 17 0 0.00 0.00 - no Open
1080 5.339181214027544 -0.929592 -23.1893 10 16 0 0.00 0.00 - no Open
583 5.630799113426268 -1.04133 -26.5489 9 21 0 0.00 0.00 - no Open
1961 4.909886224393236 -0.90485 -24.7932 3 17 0 0.00 0.00 - yes Open
2064 6.977560368249202 -0.921564 -27.0509 5 15 10 0.50 0.00 - yes Current
1190 7.1157636358790235 -0.674942 -19.2002 6 16 0 0.00 0.00 - yes Open
582 8.463256946645911 -0.924977 -28.5631 11 15 0 0.00 0.00 - yes Open
1079 9.918314688126125 -0.901996 -22.4202 13 16 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -27.051kcal/mol
Ligand efficiency (LE) -0.9017kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -8.698
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 30HA

Physicochemical properties

Molecular weight 428.5Da
Lipinski: ≤ 500 Da
LogP (cLogP) 4.30
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 11.23kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 88.56kcal/mol
Minimised FF energy 77.33kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.